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| | 2'-MECCPA Basic information |
| Product Name: | 2'-MECCPA | | Synonyms: | 2'-MECCPA;2-CHLORO-N-CYCLOPENTYL-2'-METHYLADENOSINE;-MeCCPA;2'-Chloro-N6-cyclopentyl-2'-methyl adenosine;Adenosine, 2-chloro-N-cyclopentyl-2'-C-methyl-;2' MeCCPA,2'MeCCPA;2'-MeCCPA;2-Chloro-N-cyclopentyl-2'-Methyladenosine | | CAS: | 205171-12-6 | | MF: | C16H22ClN5O4 | | MW: | 383.83 | | EINECS: | | | Product Categories: | | | Mol File: | 205171-12-6.mol |  |
| | 2'-MECCPA Chemical Properties |
| Boiling point | 643.3±65.0 °C(Predicted) | | density | 1.76±0.1 g/cm3(Predicted) | | storage temp. | Store at +4°C | | solubility | Soluble to 25 mM in DMSO | | form | Powder | | pka | 13.13±0.70(Predicted) |
| | 2'-MECCPA Usage And Synthesis |
| Uses | 2''-?MeCCPA is an inhibitor of forskolin-stimulated adenylyl cyclase. It is also a selective A1 adenosine receptor agonist. | | Definition | ChEBI: 2-[2-chloro-6-(cyclopentylamino)-9-purinyl]-5-(hydroxymethyl)-3-methyloxolane-3,4-diol is a purine nucleoside. | | Biological Activity | Potent and highly selective agonist at A 1 adenosine receptors (K i values are 3.3, 9580, 37600 and 1150 nM for human recombinant A 1 , A 2A , A 2B and A 3 receptors respectively). Acts as a full agonist; inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC 50 value of 13.1 nM. | | storage | Store at +4°C |
| | 2'-MECCPA Preparation Products And Raw materials |
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