| Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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| Tel: |
821-50328103-801 18930552037 |
| Email: |
3bsc@sina.com |
| Products Intro: |
Product Name:Telenzepine dihydrochloride;4,9-Dihydro-3-Methyl-4-[(4-Methyl-1-piperazinyl)acetyl]-10H-thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride
CAS:147416-96-4
Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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| Company Name: |
BOC Sciences
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| Tel: |
1-631-485-4226; 16314854226 |
| Email: |
info@bocsci.com |
| Products Intro: |
Product Name:Telenzepine dihydrochloride
CAS:147416-96-4
Remarks:Telenzepine dihydrochloride is a selective and high affinity muscarinic M1 receptor antagonist (Ki = 0.94 nM). Telenzepine was demonstrated ability to inhibit gastric acid secretion.
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| | TELENZEPINE DIHYDROCHLORIDE Basic information |
| Product Name: | TELENZEPINE DIHYDROCHLORIDE | | Synonyms: | 4,9-DIHYDRO-3-METHYL-4-[(4-METHYL-1-PIPERAZINYL)ACETYL]-10H-THIENO[3,4-B][1,5] BENZODIAZEPIN-10-ONE DIHYDROCHLORIDE;TELENZEPINE DIHYDROCHLORIDE;TELENZEPINE DIHYDROCHLORIDE SELECTIVE M1 MUSCARIN;4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride;Telenzepine dihydrochloide;Telenzepine hydrate dihydrochloride;4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H);JTQJFSQQHGPLOX-UHFFFAOYSA-N | | CAS: | 147416-96-4 | | MF: | C19H22N4O2S | | MW: | 370.47 | | EINECS: | | | Product Categories: | Acetylcholine receptor | | Mol File: | 147416-96-4.mol |  |
| | TELENZEPINE DIHYDROCHLORIDE Chemical Properties |
| storage temp. | Store at RT | | solubility | H2O: >10 mg/mL | | form | solid | | color | white | | Water Solubility | Soluble to 100 mM in water |
| | TELENZEPINE DIHYDROCHLORIDE Usage And Synthesis |
| Uses | Telenzepine dihydrochloride is a potent and selective muscarnic receptor antagonist. | | Uses | Telenzepine dihydrochloride hydrate was used to study M1 muscarinic receptor-mediated signaling in juvenile rat hippocampus and rat urinary bladder. | | Uses | Antiulcerative;M1 muscarinic antagonist | | Biological Activity | Selective high affinity muscarinic M 1 receptor antagonist (K i = 0.94 nM). Inhibits gastric acid secretion. | | Biochem/physiol Actions | Telenzepine is an analog of pirenzepine and inhibits the secretion of gastric acid. It is an antagonist to M1-receptor and targets the oxyntic gastric glands and the salivary glands. | | storage | Desiccate at RT |
| | TELENZEPINE DIHYDROCHLORIDE Preparation Products And Raw materials |
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