| Identification | Back Directory | [Name]
L-Valinamide, N-(3,5-dimethylbenzoyl)-4-(5-isoxazolyl)-N-methyl-D-phenylalanyl-N-(butylsulfonyl)- | [CAS]
173189-01-0 | [Synonyms]
IRL3630
IRL-3630
IRL 3630
L-Valinamide, N-(3,5-dimethylbenzoyl)-4-(5-isoxazolyl)-N-methyl-D-phenylalanyl-N-(butylsulfonyl)- | [Molecular Formula]
C31H40N4O6S | [MOL File]
173189-01-0.mol | [Molecular Weight]
596.74 |
| Hazard Information | Back Directory | [Uses]
IRL-3630 (Compound 3) is an ETA/ETB antagonist (Ki: 1.9 and 1.2 nM)[1]. | [References]
[1] Sakaki J, et al. Stereoselective synthesis of a novel and bifunctional endothelin antagonist, IRL 3630. Bioorg Med Chem Lett. 1998 Aug 18;8(16):2247-52. DOI:10.1016/s0960-894x(98)00388-6 |
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