Muscarinic toxin 1

Muscarinic toxin 1 Struktur
CAS-Nr.
Englisch Name:
Muscarinic toxin 1
Synonyma:
MT1;MTX1;MEL-1A-R;MT1; MT 1;MUSCARINIC TOXIN 1;Mel1a melatonin receptor;Anti-MTR1A antibody produced in rabbit;Anti-MTNR1A antibody produced in rabbit;Muscarinic Toxin-1 from Dendroaspis angusticeps venom;LEU-THR-CYS-VAL-THR-SER-LYS-SER-ILE-PHE-GLY-ILE-THR-THR-GLU-ASN-CYS-PRO-ASP-GLY-GLN-ASN-LEU-CYS-PHE-LYS-LYS-TRP-TYR-TYR-ILE-VAL-PRO-ARG-TYR-SER-ASP-ILE-THR-TRP-GLY-CYS-ALA-ALA-THR-CYS-PRO-LYS-PRO-THR-ASN-VAL-ARG-GLU-THR-ILE-ARG-CYS-CYS-GLU-THR-ASP-LYS-CYS-ASN-GLU
CBNumber:
CB3392337
Summenformel:
Molgewicht:
0
MOL-Datei:
Mol file

Muscarinic toxin 1 Eigenschaften

storage temp. 
−20°C
Aggregatzustand
lyophilized powder

Sicherheit

WGK Germany  3

Muscarinic toxin 1 Chemische Eigenschaften,Einsatz,Produktion Methoden

Biologische Funktion

Muscarinic toxin 1 has non-competitive interactions with adrenergic and muscarinic receptors. Binds to alpha-2b (ADRA2B) (IC50=2.3 nM), alpha-1a (ADRA1A), alpha-1b (ADRA1B) and alpha-2c (ADRA2C) adrenergic receptors. Reversibly binds to the M1 (CHRM1) muscarinic acetylcholine receptor, probably through interaction with the orthosteric site. Also has slightly weaker effects on M3 (CHRM3) and M4 (CHRM4) receptors. The order of potency is ADRA2B>>CHRM1>ADRA1A>ADRA1B>ADRA2C/CHRM4 (PubMed:24793485).

Advantages

Muscarinic toxins isolated from the venom of Dendroaspis snakes may interact with a high affinity, large selectivity and various functional properties with muscarinic receptors.

Muscarinic toxin 1 Upstream-Materialien And Downstream Produkte

Upstream-Materialien

Downstream Produkte


Muscarinic toxin 1 Anbieter Lieferant Produzent Hersteller Vertrieb Händler.

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  • Anti-MTNR1A antibody produced in rabbit
  • Anti-MTR1A antibody produced in rabbit
  • LEU-THR-CYS-VAL-THR-SER-LYS-SER-ILE-PHE-GLY-ILE-THR-THR-GLU-ASN-CYS-PRO-ASP-GLY-GLN-ASN-LEU-CYS-PHE-LYS-LYS-TRP-TYR-TYR-ILE-VAL-PRO-ARG-TYR-SER-ASP-ILE-THR-TRP-GLY-CYS-ALA-ALA-THR-CYS-PRO-LYS-PRO-THR-ASN-VAL-ARG-GLU-THR-ILE-ARG-CYS-CYS-GLU-THR-ASP-LYS-CYS-ASN-GLU
  • MT1
  • MUSCARINIC TOXIN 1
  • MTX1
  • Muscarinic Toxin-1 from Dendroaspis angusticeps venom
  • MEL-1A-R
  • Mel1a melatonin receptor
  • MT1; MT 1
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