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Epitinib (succinate)

CAS No.
2252334-12-4
Chemical Name:
Epitinib (succinate)
Synonyms
Epitinib (succinate)
CBNumber:
CB010222443
Molecular Formula:
C28H32N6O6
Molecular Weight:
548.6
MDL Number:
MOL File:
2252334-12-4.mol
MSDS File:
SDS
Last updated:2026-07-27 17:00:41

Epitinib (succinate) Properties

storage temp. Store at -20°C
form Solid
color White to light yellow
FDA UNII 2138WW3F3R

Epitinib (succinate) price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Biosynth CQD33412 Epitinib succinate 2252334-12-4 25mg $1382.75 2026-06-04 Buy
Biosynth CQD33412 Epitinib succinate 2252334-12-4 50mg $1923.5 2026-06-04 Buy
ChemScene CS-0188812 Epitinib succinate 99.01% 2252334-12-4 5mg $314 2026-06-04 Buy
ChemScene CS-0188812 Epitinib succinate 99.01% 2252334-12-4 10mg $471 2026-06-04 Buy
ChemScene CS-0188812 Epitinib succinate 99.01% 2252334-12-4 25mg $848 2026-06-04 Buy
Product number Packaging Price Buy
CQD33412 25mg $1382.75 Buy
CQD33412 50mg $1923.5 Buy
CS-0188812 5mg $314 Buy
CS-0188812 10mg $471 Buy
CS-0188812 25mg $848 Buy

Epitinib (succinate) Chemical Properties, Uses, Production

Uses

Epitinib succinate is an orally active and selective epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI) designed for optimal brain penetration. Epitinib succinate can be used for the research of cancer[1][2]. Epitinib (succinate) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

References

[1] Zhou et al. The safety profile of a selective EGFR TKI epitinib (HMPL-813) in patients with advanced solid tumors and preliminary clinical efficacy in EGFRm+ NSCLC patients with brain metastasis. Journal of Clinical Oncology 2016 34:15_suppl, e20502-e20502
[2] Zhou et al. Phase I study of the safety and pharmacokinetics of epitinib, an oral EGFR tyrosine kinase inhibitor, in patients with advanced solid tumors. Journal of Clinical Oncology 2013 31:15_suppl, e19042-e19042

Epitinib (succinate) Preparation Products And Raw materials

Raw materials

Preparation Products

Epitinib (succinate) Suppliers

Global Suppliers ( 14)
Supplier Tel Email Country ProdList Advantage
BOC Sciences 16314854226; +8616314854226 inquiry@bocsci.com United States 19852 58
TargetMol Chemicals Inc. +1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
Jinan Jiuli Biotechnology Co. , Ltd. 15865264761 486064515@qq.com China 5000 58
Shanghai Yifei Biotechnology Co. , Ltd. 021-65675885 18964387627 customer_service@efebio.com China 11963 58
Beijing Boorsen Biotechnology Co., Ltd 400-901-9800 18611424007 cis@bioss.com.cn China 9185 58
RD International Technology Co., Limited 18024082417 market@ubiochem.com China 9831 58
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29873 58
Shanghai Amole Biotechnology Co., Ltd. 13370042665 18916960931 2596183085@qq.com China 17234 58
Aladdin Scientific tp@aladdinsci.com United States 50068 58

View Latest Price from Epitinib (succinate) manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Epitinib succinate pictures 2026-07-27 Epitinib succinate
2252334-12-4
$69.00-173.00 99.79% 10g TargetMol Chemicals Inc.

Epitinib (succinate) Spectrum

Epitinib (succinate) 2252334-12-4