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GSK 2239633A

GSK 2239633A Structure
GSK 2239633A structure
CAS No.
1240516-71-5
Chemical Name:
GSK 2239633A
Synonyms
GSK 2239633A;GSK2239633A, 10 mM in DMSO;GSK-2239633A,inhibit,Inhibitor,CC chemokine receptor,CCR,GSK2239633A;Propanamide, N-[[3-[[3-[[(5-chloro-2-thienyl)sulfonyl]amino]-4-methoxy-1H-indazol-1-yl]methyl]phenyl]methyl]-2-hydroxy-2-methyl-;N-[(3-{[3-{[(5-Chloro-2-thienyl)sulfonyl]amino}-4-(methyloxy)-1H-indazol-1-yl]methyl}phenyl)methyl]-2-hydroxy-2-methylpropanamide
CBNumber:
CB14189083
Molecular Formula:
C24H25ClN4O5S2
Molecular Weight:
549.06
MDL Number:
MFCD30533311
MOL File:
1240516-71-5.mol
Last updated:2025-09-30 18:11:34
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GSK 2239633A Properties

Density 1.45±0.1 g/cm3(Predicted)
storage temp. Store at -20°C
solubility DMSO:152.46(Max Conc. mg/mL);277.67(Max Conc. mM)
pka 7.03±0.30(Predicted)
form Solid
color White to off-white
InChIKey YTEVTHHGQMUPHC-UHFFFAOYSA-N
SMILES C(NCC1=CC=CC(CN2C3=C(C(OC)=CC=C3)C(NS(C3SC(Cl)=CC=3)(=O)=O)=N2)=C1)(=O)C(O)(C)C
FDA UNII 07ODS257BP

GSK 2239633A price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Tocris 7071 GSK2239633A ≥98%(HPLC) 1240516-71-5 50 $965 2021-12-16 Buy
TRC G797595 GSK2239633A 1240516-71-5 10mg $2310 2021-12-16 Buy
TRC G797595 GSK2239633A 1240516-71-5 1mg $290 2021-12-16 Buy
ChemScene CS-0018178 GSK2239633A 99.77% 1240516-71-5 5mg $550 2021-12-16 Buy
ChemScene CS-0018178 GSK2239633A 99.77% 1240516-71-5 10mg $850 2021-12-16 Buy
Product number Packaging Price Buy
7071 50 $965 Buy
G797595 10mg $2310 Buy
G797595 1mg $290 Buy
CS-0018178 5mg $550 Buy
CS-0018178 10mg $850 Buy

GSK 2239633A Chemical Properties,Uses,Production

Uses

GSK 2239633A, is an allosteric antagonist of human CCR4.

in vivo

Following intravenous dosing, plasma GSK2239633A displays rapid, bi-phasic distribution and slow terminal elimination (t1/2: 13.5 hours), suggesting that GSK2239633A is a low to moderate clearance drug. Following oral dosing, blood levels of GSK2239633A reach Cmax rapidly (median tmax: 1.0-1.5 hours). Estimated GSK2239633A bioavailability is low with a maximum value determined of only 16%[1]. GSK2239633A (Compound 9) demonstrates good pharmacokinetic data in preclinical animal studies (bioavailability in rats and beagle dogs 85% and 97% respectively)[3].

IC 50

[125I]-TARC-CCR4: 7.96 (pIC50)

storage

Store at -20°C

GSK 2239633A Preparation Products And Raw materials

Raw materials

Preparation Products

GSK 2239633A Suppliers

Global( 32)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. 		+1-781-999-5354; +17819995354 marketing@targetmol.com United States 32432 58
InvivoChem 		+1-708-310-1919 +1-13798911105 sales@invivochem.cn United States 6391 58
TargetMol Chemicals Inc. 		+1-781-999-5354; support@targetmol.com United States 39031 58
Wuhan Topule Biopharmaceutical Co., Ltd 		+8618327326525 masar@topule.com China 8467 58
Aladdin Scientific 		tp@aladdinsci.com United States 57505 58
Amadis Chemical Company Limited 		571-89925085 sales@amadischem.com China 131957 58
Hangzhou ChangCun Biotechnology Co., Ltd. 0571-; 13567100326 158848739@qq.com China 108 50
Shanghai YuanYe Biotechnology Co., Ltd. 021-61312847; 18021002903 3008007409@qq.com China 71826 60
ShangHai Biochempartner Co.,Ltd 177-54423994 17754423994 2853530910@QQ.com China 8000 62
Aikon International Limited 025-58851090 15955137747 sales01@aikonchem.com China 15949 58
Supplier Advantage
TargetMol Chemicals Inc. 		58
InvivoChem 		58
TargetMol Chemicals Inc. 		58
Wuhan Topule Biopharmaceutical Co., Ltd 		58
Aladdin Scientific 		58
Amadis Chemical Company Limited 		58
Hangzhou ChangCun Biotechnology Co., Ltd. 50
Shanghai YuanYe Biotechnology Co., Ltd. 60
ShangHai Biochempartner Co.,Ltd 62
Aikon International Limited 58

View Lastest Price from GSK 2239633A manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
GSK2239633A pictures 2025-09-30 GSK2239633A
1240516-71-5
 US $32.00-127.00 / mg 99.82% 10g TargetMol Chemicals Inc.
GSK2239633A pictures 2025-09-30 GSK2239633A
1240516-71-5
 US $32.00-127.00 / mg 99.82% 10g TargetMol Chemicals Inc.
  • GSK2239633A pictures
  • GSK2239633A
    1240516-71-5
  • US $32.00-127.00 / mg
  • 99.82%
  • TargetMol Chemicals Inc.
  • GSK2239633A pictures
  • GSK2239633A
    1240516-71-5
  • US $32.00-127.00 / mg
  • 99.82%
  • TargetMol Chemicals Inc.

1240516-71-5(GSK 2239633A)Related Search:

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MethanesulfonaMide, N-[5-[4-[5-[[(2R,6S)-2,6-diMethyl-4-Morpholinyl]Methyl]-2-oxazolyl]-1H-indazol-6-yl]-2-Methoxy-3-pyridinyl]-, rel- GSK2636771 GSK-2881078 gsk2200150a GSK-2018682
Lp-PLA2 -IN-1 GSK-3326595

1of3

GSK 2239633A Propanamide, N-[[3-[[3-[[(5-chloro-2-thienyl)sulfonyl]amino]-4-methoxy-1H-indazol-1-yl]methyl]phenyl]methyl]-2-hydroxy-2-methyl- GSK-2239633A,inhibit,Inhibitor,CC chemokine receptor,CCR,GSK2239633A N-[(3-{[3-{[(5-Chloro-2-thienyl)sulfonyl]amino}-4-(methyloxy)-1H-indazol-1-yl]methyl}phenyl)methyl]-2-hydroxy-2-methylpropanamide GSK2239633A, 10 mM in DMSO 1240516-71-5 C24H25ClN4O5S2