Chinese Japanese Germany Korea
ChemicalBook >> CAS DataBase List >>Befloxatone

Befloxatone

Befloxatone Structure
Befloxatone structure
CAS No.
134564-82-2
Chemical Name:
Befloxatone
Synonyms
503;MD-370;MD370503;MD-370503;MD 370503;Befloxatone;(R)-5-(methoxymethyl)-3-(4-((R)-4,4,4-trifluoro-3-hydroxybutoxy)phenyl)oxazolidin-2-one;2-Oxazolidinone, 5-(methoxymethyl)-3-[4-[(3R)-4,4,4-trifluoro-3-hydroxybutoxy]phenyl]-, (5R)-
CBNumber:
CB2874979
Molecular Formula:
C15H18F3NO5
Molecular Weight:
349.3
MDL Number:
MFCD00871024
MOL File:
134564-82-2.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-05-11 19:39:08
Request For Quotation

Befloxatone Properties

Melting point 101°
alpha D20 -11.5° (c = 1 in methylene chloride)
Boiling point 447.3±45.0 °C(Predicted)
Density 1.326±0.06 g/cm3(Predicted)
pka 12.13±0.20(Predicted)
FDA UNII 4H75PAD8M3

Befloxatone price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
American Custom Chemicals Corporation API0010777 BEFLOXATONE 95.00% 134564-82-2 5MG $501.2 2021-12-16 Buy
Product number Packaging Price Buy
API0010777 5MG $501.2 Buy

Befloxatone Chemical Properties,Uses,Production

Uses

Befloxatone is a selective and reversible inhibitor of monoamine oxidase A. A third line agent for the treatment of resistant depression.

in vivo

Befloxatone (0.75 mg/kg; i.p.; single dose) increases tissue levels of monoamines and decreases levels of their deaminating metabolites in rats[1].
Befloxatone (1 mg/kg; i.p.; single dose) induces elevated levels of dopamine and corticonorepinephrine in the extracellular striatum of rats, but not elevates levels of corticoserotonin[1].
Befloxatone (0.03-0.3 mg/kg; p.o.; single dose) effectively inhibits the firing rate of serotonergic neurons and partially reduces the firing of norepinephric neurons, but had no effect on the firing of dopaminergic neurons in rats[1].
Befloxatone (1.5 mg/kg; p.o.; single dose) does not enhance the pressor effect of the central active dose of oral tyramine and has a broad safety profile in rats[1].

IC 50

MAO-A: 4 nM (IC50); MAO-B: 300 nM (IC50)

Befloxatone Preparation Products And Raw materials

Raw materials

Preparation Products

Befloxatone Suppliers

Global( 7)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. +1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
TargetMol Chemicals Inc. 13564774135 marketing@targetmol.com United States 19950 58
Supplier Advantage
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58

View Lastest Price from Befloxatone manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Befloxatone pictures 2026-05-11 Befloxatone
134564-82-2
 $1520.00-2500.00 10g TargetMol Chemicals Inc.
  • Befloxatone pictures
  • Befloxatone
    134564-82-2
  • $1520.00-2500.00
  • TargetMol Chemicals Inc.

134564-82-2(Befloxatone)Related Search:

Methyl N-(4-methoxyphenyl)carbamate (4-Methoxy-phenyl)-carbamic acid ethyl ester 3-Phenyl-2-oxazolidinone (R)-5-(HYDROXYMETHYL)-3-METHYLOXAZOLIDIN-2-ONE 5-HYDROXYMETHYL-3-(4-METHOXYPHENYL)-2-OXAZOLIDINONE
(R)-5-(HYDROXYMETHYL)-3-PHENYLOXAZOLIDIN-2-ONE Befloxatone (R)-5-METHOXYMETHYL-2-OXAZOLIDINONE (R)-4,4,4-TRIFLUOROBUTANE-1,3-DIOL

1of2

Befloxatone (R)-5-(methoxymethyl)-3-(4-((R)-4,4,4-trifluoro-3-hydroxybutoxy)phenyl)oxazolidin-2-one 2-Oxazolidinone, 5-(methoxymethyl)-3-[4-[(3R)-4,4,4-trifluoro-3-hydroxybutoxy]phenyl]-, (5R)- MD 370503 MD-370 MD370503 MD-370503 503 134564-82-2 C15H18F3NO5