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ChemicalBook >> CAS DataBase List >>Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Structure
Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid structure
CAS No.
500577-51-5
Chemical Name:
Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid
Synonyms
Cyclo(-RGDfK) Trifluoroacetate;Cyclo(-RGDfK) TFA, 10 mM in DMSO;Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid;Cyclo(-Arg-Gly-Asp-D-Phe-Lys) trifluoroacetate;2-((2S,5R,8S,11S)-8-(4-Aminobutyl)-5-benzyl-11-(3-guanidinopropyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentaazacyclopentadecan-2-yl)acetic acid Trifluoroacetate (1:1);2,2,2-trifluoroacetic acid--2-((2S,5R,8S,11S)-8-(4-aminobutyl)-5-benzyl-11-(3-guanidinopropyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentaazacyclopentadecan-2-yl)acetic acid (1/1)
CBNumber:
CB33367651
Molecular Formula:
C29H42F3N9O9
Molecular Weight:
717.6938896
MDL Number:
MOL File:
500577-51-5.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-07-27 17:00:41
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Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Properties

storage temp. under inert gas (nitrogen or Argon) at 2–8 °C
solubility DMSO: 100 mg/mL (139.34 mM)
form Solid
color White to off-white
Water Solubility Water: 33.33 mg/mL (46.44 mM)
Sequence Cyclo(Arg-Gly-Asp-Phe-Lys)

SAFETY

Risk and Safety Statements

Symbol(GHS)  Exclamation Mark (GHS07)
GHS07
Signal word  Warning
Hazard statements  H302-H315-H319-H335
Precautionary statements  P280-P305+P351+P338

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Biosynth FC110054 Cyclo(-Arg-Gly-Asp-D-Phe-Lys) trifluoroacetate 500577-51-5 10mg $290.4 2026-06-04 Buy
Biosynth FC110054 Cyclo(-Arg-Gly-Asp-D-Phe-Lys) trifluoroacetate 500577-51-5 25mg $680.75 2026-06-04 Buy
Biosynth FC110054 Cyclo(-Arg-Gly-Asp-D-Phe-Lys) trifluoroacetate 500577-51-5 50mg $1270.5 2026-06-04 Buy
Biosynth FC110054 Cyclo(-Arg-Gly-Asp-D-Phe-Lys) trifluoroacetate 500577-51-5 100mg $2360 2026-06-04 Buy
ChemScene CS-0102584 Cyclo(-RGDfK) TFA 99.61% 500577-51-5 5mg $151 2026-06-04 Buy
Product number Packaging Price Buy
FC110054 10mg $290.4 Buy
FC110054 25mg $680.75 Buy
FC110054 50mg $1270.5 Buy
FC110054 100mg $2360 Buy
CS-0102584 5mg $151 Buy

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Chemical Properties, Uses, Production

Uses

Cyclo(-RGDfK) TFA is a potent and selective inhibitor of the αvβ3 integrin, with an IC50 of 0.94 nM[1]. Cyclo(-RGDfK) TFA potently targets tumor microvasculature and cancer cells through the specific binding to the αvβ3 integrin on the cell surface[3].

IC 50

αvβ3: 0.94 nM (IC50)

References

[1] Simecek J, et al. Benefits of NOPO as chelator in gallium-68 peptides, exemplified by preclinical characterization of (68)Ga-NOPO-c(RGDfK). Mol Pharm. 2014 May 5;11(5):1687-95. DOI:10.1021/mp5000746
[2] Lopez-Rodriguez V, et al. Preparation and preclinical evaluation of (66)Ga-DOTA-E(c(RGDfK))2 as a potential theranostic radiopharmaceutical. Nucl Med Biol. 2015 Feb;42(2):109-14. DOI:10.1016/j.nucmedbio.2014.09.010

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Preparation Products And Raw materials

Raw materials

Preparation Products

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Suppliers

Global Suppliers ( 41)
Supplier Tel Email Country ProdList Advantage
Shanghai YuanYe Biotechnology Co., Ltd. 15026964105 2881489226@qq.com China 89667 60
Shanghai Chaolan Chemical Technology Center QQ：65489617 13301690235 Sales@ATKchemical.com China 9729 58
Amadis Chemical Company Limited 571-89925085 sales@amadischem.com China 131885 58
Hangzhou Peptidego Biotech Co.,Ltd. 0571-87213919 15967184799 Eric@peptidego.com China 7872 58
Shanghai Jizhi Biochemical Technology Co. Ltd. 021-4009004166/18616739031 18616739031 3007523370@qq.com China 40000 58
Shanghai Hongye Biotechnology Co. Ltd 400-9205774 400-920-5774 sales@glpbio.cn China 6705 58
BOC Sciences 16314854226; +8616314854226 inquiry@bocsci.com United States 19852 58
TargetMol Chemicals Inc. +1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
ChemeGen(Shanghai) Biotechnology Co.,Ltd. 18818260767 sales@chemegen.com China 11123 58
Nanchang Tianzhen Biotechnology Co., Ltd 13758194781 13173652190 522013271@qq.com China 2436 58
Supplier Advantage
Shanghai YuanYe Biotechnology Co., Ltd. 60
Shanghai Chaolan Chemical Technology Center 58
Amadis Chemical Company Limited 58
Hangzhou Peptidego Biotech Co.,Ltd. 58
Shanghai Jizhi Biochemical Technology Co. Ltd. 58
Shanghai Hongye Biotechnology Co. Ltd 58
BOC Sciences 58
TargetMol Chemicals Inc. 58
ChemeGen(Shanghai) Biotechnology Co.,Ltd. 58
Nanchang Tianzhen Biotechnology Co., Ltd 58

View Latest Price from Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Cyclo(-RGDfK) TFA pictures 2026-07-27 Cyclo(-RGDfK) TFA
500577-51-5
 $47.00-168.00 98.99% 10g TargetMol Chemicals Inc.

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Spectrum

Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid(500577-51-5)1HNMR

500577-51-5 (Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid) Related Search:

cyclo (Arg-Ala-Asp-d-Phe-Lys) N-butyl-N,N',N'-trimethylsulfamide ArgTX-48 TFA Ac-RYYRIK-NH2 TFA Fsllry-NH2 TFA
SAMβA TFA

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Cyclo (-RGDfK) 2,2,2-Trifluoroacetic acid Cyclo(-RGDfK) Trifluoroacetate 2-((2S,5R,8S,11S)-8-(4-Aminobutyl)-5-benzyl-11-(3-guanidinopropyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentaazacyclopentadecan-2-yl)acetic acid Trifluoroacetate (1:1) Cyclo(-RGDfK) TFA, 10 mM in DMSO Cyclo(-Arg-Gly-Asp-D-Phe-Lys) trifluoroacetate 2,2,2-trifluoroacetic acid--2-((2S,5R,8S,11S)-8-(4-aminobutyl)-5-benzyl-11-(3-guanidinopropyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentaazacyclopentadecan-2-yl)acetic acid (1/1) 500577-51-5