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M-2912

M-2912 structure

CAS No.: 1460285-69-1

Chemical Name:: M-2912

Synonyms: M-2912;Tankyrase-IN-5;Pyrrolo[1,2-a]pyrazin-1(2H)-one, 3-[4-(1-hydroxy-1-methylethyl)phenyl]-7-methyl-

CBNumber:: CB712397199

Molecular Formula:: C17H18N2O2

Molecular Weight:: 282.34

MDL Number:

MOL File:: 1460285-69-1.mol

TDS File:: TDS

Last updated:2026-07-27 17:00:41

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M-2912 Properties

Boiling point	442.6±45.0 °C(Predicted)
Density	1.20±0.1 g/cm3(Predicted)
pka	11.17±0.40(Predicted)

M-2912 Chemical Properties,Uses,Production

Uses

Tankyrase-IN-5 (Compound 30f), an analogue of MSC2504877 (HY-123851), is a tankyrase TNKS1 and TNKS2 inhibitor with IC50s of 2.3 nM and 7.9 nM, respectively[1].

References

[1] Buchstaller HP, et al. Optimization of a Screening Hit toward M2912, an Oral Tankyrase Inhibitor with Antitumor Activity in Colorectal Cancer Models. J Med Chem. 2021 Jul 22;64(14):10371-10392. DOI:10.1021/acs.jmedchem.1c00800

M-2912 Preparation Products And Raw materials

Raw materials

Preparation Products

M-2912 Suppliers

Global( 2)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
TargetMol Chemicals Inc.	15002134094	marketing@targetmol.cn	China	29874	58
TargetMol Chemicals Inc.	13564774135	marketing@targetmol.com	United States	19950	58

Supplier	Advantage
TargetMol Chemicals Inc.	58
TargetMol Chemicals Inc.	58

View Lastest Price from M-2912 manufacturers

Image	Update time	Product	Price	Min. Order	Purity	Supply Ability	Manufacturer
	2026-07-27	Tankyrase-IN-5 1460285-69-1				10g	TargetMol Chemicals Inc.

Tankyrase-IN-5
1460285-69-1
TargetMol Chemicals Inc.

1460285-69-1(M-2912)Related Search:

Olaparib 7,8-Dihydroxycoumarin 2-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1,3-dioxoisoindoline-5-carboxylic acid Fluzoparib RMC-7977

Pamiparib

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M-2912 Pyrrolo[1,2-a]pyrazin-1(2H)-one, 3-[4-(1-hydroxy-1-methylethyl)phenyl]-7-methyl- Tankyrase-IN-5 1460285-69-1