ChemicalBook >> CAS DataBase List >>4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole

CAS No.
863238-73-7
Chemical Name:
4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole
Synonyms
1-Trityl-1H-pyrazole-4-boronic acid pinacol ester;4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H...;4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-pyrazole;4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole;4-(tetraMethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylMethyl)-1H-pyrazole;4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylmethyl)pyrazole;4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylmethyl)-1H-pyrazole;1H-Pyrazole, 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylmethyl)-
CBNumber:
CB72470112
Molecular Formula:
C28H29BN2O2
Molecular Weight:
436.35
MDL Number:
MFCD10698507
MOL File:
863238-73-7.mol
MSDS File:
SDS
Last updated:2026-05-28 02:52:48
Product description Number Pack Size Price
4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole 073612 1.00g $347
4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole 073612 5.00g $899
4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole 97% AA004M8N 250mg $12
4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole 97% AA004M8N 1g $29
4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole 97% AA004M8N 5g $114
More product size

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole Properties

Boiling point 587.3±50.0 °C(Predicted)
Density 1.07±0.1 g/cm3 (20 ºC 760 Torr)
storage temp. under inert gas (nitrogen or Argon) at 2-8°C
pka 1.37±0.10(Predicted)
Appearance White to off-white Solid

SAFETY

Risk and Safety Statements

Symbol(GHS)  Exclamation Mark (GHS07)
GHS07
Signal word  Warning
Hazard statements  H302-H315-H319-H332-H335
Precautionary statements  P261-P280-P305+P351+P338

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole price More Price(35)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Matrix Scientific 073612 4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole 863238-73-7 1.00g $347 2026-05-18 Buy
Matrix Scientific 073612 4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole 863238-73-7 5.00g $899 2026-05-18 Buy
aablocks AA004M8N 4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole 97% 863238-73-7 250mg $12 2026-05-28 Buy
aablocks AA004M8N 4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole 97% 863238-73-7 1g $29 2026-05-28 Buy
aablocks AA004M8N 4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole 97% 863238-73-7 5g $114 2026-05-28 Buy
Product number Packaging Price Buy
073612 1.00g $347 Buy
073612 5.00g $899 Buy
AA004M8N 250mg $12 Buy
AA004M8N 1g $29 Buy
AA004M8N 5g $114 Buy

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole Chemical Properties,Uses,Production

Synthesis

4-BROMO-1-TRITYL-1H-PYRAZOLE

95162-14-4

Bis(pinacolato)diboron

73183-34-3

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole

863238-73-7

The general procedure for the synthesis of 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-1H-pyrazole from 1-trityl-4-bromopyrazole and bis(pinacolato)diboron was carried out in the following manner: under stirring conditions, 5.0 g (12.8 mmol) of 1-trityl-4-bromo-1H-pyrazole, 9.8 g (38.6 mmol, 3.0 eq.) bis(pinacolato)diboron, 1.0 g (1.3 mmol, 10 mol%) of PdCl2 (dppf), and 6.3 g (64.2 mmol, 5.0 eq.) of potassium acetate were dissolved in 30 mL of DMF and heated to react for 16 hr at 80 °C. After completion of the reaction, the mixture was diluted with water and the product was extracted with dichloromethane. The organic layer was sequentially washed with brine, dried over anhydrous sodium sulfate, and finally purified by fast chromatography to afford 5.1 g (91% yield) of the target compound 4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole.

References

[1] Patent: US2008/261975, 2008, A1. Location in patent: Page/Page column 12
[2] Journal of Organic Chemistry, 2018, vol. 83, # 5, p. 2954 - 2958
[3] Patent: US2009/82403, 2009, A1. Location in patent: Page/Page column 81
[4] Patent: US2007/105904, 2007, A1. Location in patent: Page/Page column 78-79

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole Preparation Products And Raw materials

Global( 65)Suppliers
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Capot Chemical Co.,Ltd.
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career henan chemical co
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Alchem Pharmtech,Inc.
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Antai Fine Chemical Technology Co.,Limited
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Guangzhou Yuheng Pharmaceutical Technology Co., Ltd
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Shanghai Daeyeon Chemicals Co., Ltd
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Hefei TNJ Chemical Industry Co.,Ltd.
+86-0551-65418684 +86-18949823763 sales@tnjchem.com China 25356 58
Coresyn Pharmatech Co., Ltd.
+86-571-86626709 +86-18157142896 cbc@coresyn.com China 9984 58
Jilin Chinese Academy of Sciences-yanshen Technology
18143011203 info@chemextension.com China 42056 58
Aladdin Scientific
tp@aladdinsci.com United States 57505 58

View Lastest Price from 4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole pictures 2019-07-06 4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole
863238-73-7
$1.00 1KG 98%-100% 1 Career Henan Chemical Co

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole Spectrum

4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H-pyrazole 4-(tetraMethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylMethyl)-1H-pyrazole 1-Trityl-1H-pyrazole-4-boronic acid pinacol ester 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-trityl-pyrazole 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylmethyl)pyrazole 1H-Pyrazole, 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylmethyl)- 4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1-trityl-1H... 4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1-(triphenylmethyl)-1H-pyrazole 863238-73-7 C28H29BN2O2