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Veldoreotide

Veldoreotide Structure
Veldoreotide structure
CAS No.
252845-37-7
Chemical Name:
Veldoreotide
Synonyms
DG-3173;Veldoreotide;ABFNTRQPWNXUHA-UHFFFAOYSA-N;Glycinamide, N-(4-amino-1-oxobutyl)-L-phenylalanyl-L-tryptophyl-D-tryptophyl-L-lysyl-L-threonyl-L-phenylalanyl-N2-(3-carboxypropyl)-, (7→1)-lactam
CBNumber:
CB73159915
Molecular Formula:
C60H74N12O10
Molecular Weight:
1123.30396
MDL Number:
MFCD28964044
MOL File:
252845-37-7.mol
TDS File:
TDS
Last updated:2026-04-24 14:58:35
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Veldoreotide Properties

Boiling point 1527.8±65.0 °C(Predicted)
Density 1.226±0.06 g/cm3(Predicted)
pka 13.23±0.70(Predicted)
FDA UNII 1Z83587HBN

Veldoreotide Chemical Properties, Uses, Production

Uses

Veldoreotide (DG3173) a somatostatin analogue, binds to and activate the somatostatin receptors (SSTR) 2, 4, and 5. Veldoreotide inhibits growth hormone (GH) secretion in adenomas compared with Octreotide (HY-P0036). Veldoreotide has the potential to be used as pain modulating agent[1]

IC 50

SSTR2: 37.6 nM (EC50); SSTR3: 31.3 nM (EC50); SSTR4: 10.5 nM (EC50)

References

[1] Dasgupta P, et al. Pharmacological Characterization of Veldoreotide as a Somatostatin Receptor 4 Agonist. Life (Basel). 2021 Oct 12;11(10):1075. DOI:10.3390/life11101075
[2] Plckinger U, et al. DG3173 (somatoprim), a unique somatostatin receptor subtypes 2-, 4- and 5-selective analogue, effectively reduces GH secretion in human GH-secreting pituitary adenomas even in Octreotide non-responsive tumours. Eur J Endocrinol. 2012 Feb;166(2):223-34. DOI:10.1530/EJE-11-0737

Veldoreotide Preparation Products And Raw materials

Raw materials

Preparation Products

Veldoreotide Suppliers

Global Suppliers ( 5)
Supplier Tel Email Country ProdList Advantage
Shanghai YuanYe Biotechnology Co., Ltd. 15026964105 2881489226@qq.com China 89667 60
Hangzhou Peptidego Biotech Co.,Ltd. 0571-87213919 15967184799 Eric@peptidego.com China 7872 58
Hubei Weideli Chemical Reagent Co., Ltd. 15871722230 15871722230@163.com China 4440 58
Hangzhou Sinoda Pharmaceutical Technology Co. LTD 0571-87213919 17306812703 3007955328@qq.com China 7446 58
Fuan Bio 15002819872 2845971812@qq.com China 2103 58
Supplier Advantage
Shanghai YuanYe Biotechnology Co., Ltd. 60
Hangzhou Peptidego Biotech Co.,Ltd. 58
Hubei Weideli Chemical Reagent Co., Ltd. 58
Hangzhou Sinoda Pharmaceutical Technology Co. LTD 58
Fuan Bio 58

252845-37-7 (Veldoreotide) Related Search:

Pasireotide Lanreotide acetate Cyclo(7-aminoheptanoyl-Phe-D-Trp-Lys-Thr[Bzl]) DOTA-NOC, DOTA-[Nal3]-octreotide D-Tyrosinamide, 4-chloro-N-[2-[4,7,10-tris(carboxymethyl)-1,4,7,10-tetraazacyclododec-1-yl]acetyl]-L-phenylalanyl-D-cysteinyl-4-[[[(4S)-hexahydro-2,6-dioxo-4-pyrimidinyl]carbonyl]amino]-L-phenylalanyl-4-[(aminocarbonyl)amino]-D-phenylalanyl-L-lysyl-L-threonyl-L-cysteinyl-, cyclic (2→7)-disulfide
Octreotide acetate

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ABFNTRQPWNXUHA-UHFFFAOYSA-N Glycinamide, N-(4-amino-1-oxobutyl)-L-phenylalanyl-L-tryptophyl-D-tryptophyl-L-lysyl-L-threonyl-L-phenylalanyl-N2-(3-carboxypropyl)-, (7→1)-lactam Veldoreotide DG-3173 252845-37-7