Boc-D-Azetidine-2-carboxylic acid
- CAS No.
- 228857-58-7
- Chemical Name:
- Boc-D-Azetidine-2-carboxylic acid
- Synonyms
- (R)-1-(tert-butoxycarbonyl)azetidine-2-carboxylic acid;(2R)-1-tert-Butoxycarbonylazetidine-2-carboxylic acid;Boc-D-Aze-OH;(R)-1-Boc-azetidine-2-car...;(R)-N-Boc-azetodome carboxylic;Boc-D-Azetidine-2-carboxylic acid;N-Boc-R-2-Azetidinecarboxylic acid;1-Boc-D-azetidine-2-carboxylic acid;Boc-(R)-azetidine-2-carboxylic acid;(R)-N-Boc-azetidine carboxylic acid
- CBNumber:
- CB8966476
- Molecular Formula:
- C9H15NO4
- Molecular Weight:
- 201.22
- MDL Number:
- MFCD01320888
- MOL File:
- 228857-58-7.mol
- MSDS File:
- SDS
| Product description | Number | Pack Size | Price |
| BOC-D-AZETIDINE-2-CARBOXYLIC ACID 95% | SC3761 | 1G | $29 |
| BOC-D-AZETIDINE-2-CARBOXYLIC ACID 95% | SC3761 | 5G | $119 |
| BOC-D-AZETIDINE-2-CARBOXYLIC ACID 95% | SC3761 | 25G | $399 |
| (R)-Azetidine-1,2-dicarboxylic acid 1-tert-butyl ester 97% | OR309021 | 250mg | $21 |
| (R)-Azetidine-1,2-dicarboxylic acid 1-tert-butyl ester 97% | OR309021 | 1g | $29 |
| More product size | |||
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H302-H315-H319-H335 |
| Precautionary statements | P261-P305+P351+P338 |
| Risk Statements | 36/37/38 |
| Safety Statements | 26-36 |
| HS Code | 29339900 |
Boc-D-Azetidine-2-carboxylic acid price More Price(61)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| AstaTech | SC3761 | BOC-D-AZETIDINE-2-CARBOXYLIC ACID 95% | 228857-58-7 | 1G | $29 | 2026-04-30 | Buy |
| AstaTech | SC3761 | BOC-D-AZETIDINE-2-CARBOXYLIC ACID 95% | 228857-58-7 | 5G | $119 | 2026-04-30 | Buy |
| AstaTech | SC3761 | BOC-D-AZETIDINE-2-CARBOXYLIC ACID 95% | 228857-58-7 | 25G | $399 | 2026-04-30 | Buy |
| Apolloscientific | OR309021 | (R)-Azetidine-1,2-dicarboxylic acid 1-tert-butyl ester 97% | 228857-58-7 | 250mg | $21 | 2026-06-04 | Buy |
| Apolloscientific | OR309021 | (R)-Azetidine-1,2-dicarboxylic acid 1-tert-butyl ester 97% | 228857-58-7 | 1g | $29 | 2026-06-04 | Buy |
Boc-D-Azetidine-2-carboxylic acid Chemical Properties,Uses,Production
Chemical Properties
White powder
Uses
1,2-Azetidinedicarboxylic Acid 1-(1,1-Dimethylethyl) Ester, is an useful intermediate in the synthesis of pharmaceutical compounds including inhibitors and receptor Antagonists. It can be used in the synthesis of polypeptides.
Synthesis
24424-99-5
7729-30-8
228857-58-7
To a mixed solution of (R)-azetidine-2-carboxylic acid (20 g, 200 mmol), water (200 mL) and dioxane (200 mL) was slowly added dropwise a solution of di-tert-butyl dicarbonate (Boc2O) in dioxane (100 mL) at 0 °C. After the dropwise addition was completed, the reaction mixture was stirred at room temperature for 1 hour. After the reaction was complete, the mixture was concentrated and ether (200 mL) and water (200 mL) were added to the residue. The aqueous layer was acidified to pH 3-4 with 2N hydrochloric acid and then extracted with ethyl acetate (200 mL). The organic layers were combined, dried over anhydrous sodium sulfate and concentrated to give (R)-N-BOC-azetidine-2-carboxylic acid (40 g) in quantitative yield.LRMS (M-100 + H*) m/z 102.1.
References
[1] Patent: WO2008/16643, 2008, A2. Location in patent: Page/Page column 257
[2] Journal of Medicinal Chemistry, 1998, vol. 41, # 4, p. 407 - 412
[3] Patent: US6133253, 2000, A
Boc-D-Azetidine-2-carboxylic acid Preparation Products And Raw materials
Raw materials
Preparation Products
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Capot Chemical Co.,Ltd. | +86-（0）57185586718 +86-13336195806 | sales@capot.com | China | 29626 | 60 |
| Chembon Pharmaceutical Co., Ltd. | +86-28-8425-2981 | CHINA | 722 | 55 | |
| Alchem Pharmtech,Inc. | 8485655694 | sales@alchempharmtech.com | United States | 63645 | 58 |
| CONIER CHEM AND PHARMA LIMITED | sales@conier.com | China | 49906 | 58 | |
| career henan chemical co | +86-0371-86658258 | factory@coreychem.com | China | 29780 | 58 |
| Guangzhou Yuheng Pharmaceutical Technology Co., Ltd | +8613580539051 | joe@yuhengpharm.com | CHINA | 21135 | 58 |
| GL Biochem (Shanghai) Ltd. | +86-021-61263370 +86-18901917034 | CHINA | 3904 | 58 | |
| Dayang Chem (Hangzhou) Co.,Ltd. | +86-0571-88938639 17705817739 | info@dycnchem.com | China | 52693 | 58 |
| Hefei TNJ Chemical Industry Co.,Ltd. | +86-0551-65418684 +86-18949823763 | sales@tnjchem.com | China | 25333 | 58 |
| HANGZHOU LEAP CHEM CO., LTD. | +86-571-87711850 +8619957148339 | market18@leapchem.com | China | 24569 | 58 |
View Lastest Price from Boc-D-Azetidine-2-carboxylic acid manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2026-07-24 | Boc-D-Azetidine-2-carboxylic acid
228857-58-7
|
1kg | 98 | 1000kgs | Shaanxi Dideu New Materials Co. Ltd | ||
 |
2022-01-27 | Boc-d-azetidine-2-carboxylic acid
228857-58-7
|
1KG | 97.2% | 100 tons | Honest Joy Holdings Limited | ||
 |
2020-01-10 | Boc-D-Azetidine-2-carboxylic acid
228857-58-7
|
1KG | 98%; 99% | 500g;1kg； 25kg | Career Henan Chemical Co |
-
- Boc-D-Azetidine-2-carboxylic acid
228857-58-7
- $0.00
- 98
- Shaanxi Dideu New Materials Co. Ltd
-
- Boc-d-azetidine-2-carboxylic acid
228857-58-7
- $0.00
- 97.2%
- Honest Joy Holdings Limited
-
- Boc-D-Azetidine-2-carboxylic acid
228857-58-7
- $0.01
- 98%; 99%
- Career Henan Chemical Co
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