Salvinorin A Carbamate
- CAS No.
- 858345-57-0
- Chemical Name:
- Salvinorin A Carbamate
- Synonyms
- Salvinorin A Carbamate;(2S,4aR,6aR,7R,9S,10aS,10bR)-9-[(aminocarbonyl)oxy]-2-(3-furanyl)dodecahydro-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylicacid,methylester;Methyl (2S,4aR,6aR,7R,9S,10aS,10Br)-9-carbamoyloxy-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-2,4a,5,6,7,8,9,10a-octahydro-1H-benzo[f ]isochromene-7-carboxylate;2H-Naphtho[2,1-c]pyran-7-carboxylic acid, 9-[(aminocarbonyl)oxy]-2-(3-furanyl)dodecahydro-6a,10b-dimethyl-4,10-dioxo-, methyl ester, (2S,4aR,6aR,7R,9S,10aS,10bR)-
- CBNumber:
- CB94666845
- Molecular Formula:
- C22H27NO8
- Molecular Weight:
- 433.45
- MDL Number:
- MOL File:
- 858345-57-0.mol
- MSDS File:
- SDS
Salvinorin A Carbamate price More Price(10)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 22245 | Salvinorin A Carbamate ≥90% | 858345-57-0 | 500μg | $107 | 2026-04-30 | Buy |
| Cayman Chemical | 22245 | Salvinorin A Carbamate ≥90% | 858345-57-0 | 1mg | $203 | 2026-04-30 | Buy |
| Cayman Chemical | 22245 | Salvinorin A Carbamate ≥90% | 858345-57-0 | 5mg | $845 | 2026-04-30 | Buy |
| Biosynth | IJB34557 | Methyl (2S,4aR,6aR,7R,9S,10aS,10Br)-9-carbamoyloxy-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-2,4a,5,6,7,8,9,10a-octahydro-1H-benzo[f ]isochromene-7-carboxylate | 858345-57-0 | 5mg | $1428.85 | 2026-06-04 | Buy |
| Biosynth | IJB34557 | Methyl (2S,4aR,6aR,7R,9S,10aS,10Br)-9-carbamoyloxy-2-(furan-3-yl)-6a,10b-dimethyl-4,10-dioxo-2,4a,5,6,7,8,9,10a-octahydro-1H-benzo[f ]isochromene-7-carboxylate | 858345-57-0 | 10mg | $1987.9 | 2026-06-04 | Buy |
Salvinorin A Carbamate Chemical Properties, Uses, Production
Description
Salvinorin A carbamate is a potent κ-opioid receptor (KOR) full agonist that is almost as potent as salvinorin A with EC50 values of 6.2 and 4.5 nM, respectively, for activation of the human KOR to enhance binding of [35S]GTPγS. The addition of a carbamate group to salvinorin A increases biological stability by decreasing deacetylation.
Uses
Salvinorin A carbamate is an agonist for κ-opioid receptor with an EC50 of 6.2 nM and a Ki of 3.2 nM[1].
IC 50
κ Opioid Receptor/KOR: 6.2 nM (EC50)
References
[1] Béguin C, et al., Synthesis and in vitro pharmacological evaluation of salvinorin A analogues modified at C(2). Bioorg Med Chem Lett. 2005 Jun 2;15(11):2761-5. DOI:10.1016/j.bmcl.2005.03.113
Salvinorin A Carbamate Preparation Products And Raw materials
Raw materials
Preparation Products
Salvinorin A Carbamate Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Shanghai Hongye Biotechnology Co. Ltd | 400-9205774 400-920-5774 | sales@glpbio.cn | China | 6705 | 58 |
| ChemeGen(Shanghai) Biotechnology Co.,Ltd. | 18818260767 | sales@chemegen.com | China | 11123 | 58 |
| Shanghai Yifei Biotechnology Co. , Ltd. | 021-65675885 18964387627 | customer_service@efebio.com | China | 11963 | 58 |
| TargetMol Chemicals Inc. | 15002134094 | marketing@targetmol.cn | China | 29874 | 58 |
