[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate
![[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate price.](/CAS/GIF/150080-09-4.gif)
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- $33 - $6770
- Product name: [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate
- CAS: 150080-09-4
- MF: C10H23BN2O6S
- MW: 310.17
- EINECS:
- MDL Number:MFCD13194906
- Synonyms:[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate;Boronic acid, ((2R)-1-((2S)-2-amino-3-methyl-1-oxobutyl)-2-pyrrolidinyl)-, monomethanesulfonate;Unii-V8zg4Y1B51;Methanesulfonic acid ((R)-1-((S)-2-amino-3-methyl-butanoyl)pyrrolidin-2-yl)boronic acid (1:1);Talabostat mesylate;Val-boroPro mesylate;CS-1219;Talabostat-mesylate, PT-100
74 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- Adipogen Life Sciences
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Sigma-Aldrich
- Synthonix
- Tocris
- TRC
- Usbiological
Package
- 10
- 1mg
- 50
- 2mg
- 5mg
- 10mg
- 10mM(1mLinDMSO)
- 25mg
- 50mg
- 100mg
- 250mg
- 500mg
- 1.00g
- 10mM*1mLinDMSO(Solution)
- 1g
- 10mM(in 1mL DMSO)
- 5g
- 10mM*1mLinDMSO(Solid+Solvent)
- 10mM(in1mLDMSO)
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 98%
- Packaging1mg
- Price$33
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥98%(HPLC)
- Packaging2mg
- Price$44
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥95%
- Packaging5mg
- Price$54
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥95%
- Packaging10mg
- Price$91
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥95%
- Packaging25mg
- Price$209
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate
- Packaging50mg
- Price$338
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95%
- Packaging100mg
- Price$384
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95%
- Packaging250mg
- Price$616
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95%
- Packaging500mg
- Price$1024
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABJ1
- Product description[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95%
- Packaging1g
- Price$1536
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberK12105
- Product descriptionTalabostat mesylate 98%
- Packaging1G
- Price$1250
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberK12105
- Product descriptionTalabostat mesylate 98%
- Packaging100MG
- Price$330
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberK12105
- Product descriptionTalabostat mesylate 98%
- Packaging25MG
- Price$140
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberK12105
- Product descriptionTalabostat mesylate 98%
- Packaging5MG
- Price$45
- Updated2026-05-27
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CR1-3541-M010
- Product descriptionTalabostat . mesylate ≥98%(HPLC)
- Packaging10mg
- Price$70
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CR1-3541-M050
- Product descriptionTalabostat . mesylate ≥98%(HPLC)
- Packaging50mg
- Price$280
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 98% | 1mg | $33 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥98%(HPLC) | 2mg | $44 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥95% | 5mg | $54 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥95% | 10mg | $91 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate ≥95% | 25mg | $209 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate | 50mg | $338 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95% | 100mg | $384 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95% | 250mg | $616 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95% | 500mg | $1024 | 2026-05-28 | Buy |
| aablocks | AA00ABJ1 | [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate 95% | 1g | $1536 | 2026-05-28 | Buy |
| ACHEMBLOCK | K12105 | Talabostat mesylate 98% | 1G | $1250 | 2026-05-27 | Buy |
| ACHEMBLOCK | K12105 | Talabostat mesylate 98% | 100MG | $330 | 2026-05-27 | Buy |
| ACHEMBLOCK | K12105 | Talabostat mesylate 98% | 25MG | $140 | 2026-05-27 | Buy |
| ACHEMBLOCK | K12105 | Talabostat mesylate 98% | 5MG | $45 | 2026-05-27 | Buy |
| Adipogen Life Sciences | AG-CR1-3541-M010 | Talabostat . mesylate ≥98%(HPLC) | 10mg | $70 | 2026-05-06 | Buy |
| Adipogen Life Sciences | AG-CR1-3541-M050 | Talabostat . mesylate ≥98%(HPLC) | 50mg | $280 | 2026-05-06 | Buy |
Properties
Melting point :>160°C (dec.)
storage temp. :under inert gas (nitrogen or Argon) at 2–8 °C
solubility :Soluble in DMSO (up to at least 25 mg/ml)
form :solid
color :White
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChI :1S/C9H19BN2O3.CH4O3S/c1-6(2)8(11)9(13)12-5-3-4-7(12)10(14)15;1-5(2,3)4/h6-8,14-15H,3-5,11H2,1-2H3;1H3,(H,2,3,4)/t7-,8-;/m0./s1
InChIKey :OXYYOEIGQRXGPI-WSZWBAFRSA-N
SMILES :B(O)(O)[C@H]1N(CCC1)C(=O)[C@@H]([N+H3])C(C)C.[S](=O)(=O)([O-])C
storage temp. :under inert gas (nitrogen or Argon) at 2–8 °C
solubility :Soluble in DMSO (up to at least 25 mg/ml)
form :solid
color :White
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChI :1S/C9H19BN2O3.CH4O3S/c1-6(2)8(11)9(13)12-5-3-4-7(12)10(14)15;1-5(2,3)4/h6-8,14-15H,3-5,11H2,1-2H3;1H3,(H,2,3,4)/t7-,8-;/m0./s1
InChIKey :OXYYOEIGQRXGPI-WSZWBAFRSA-N
SMILES :B(O)(O)[C@H]1N(CCC1)C(=O)[C@@H]([N+H3])C(C)C.[S](=O)(=O)([O-])C
Safety Information
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| Signal word: | Warning | ||||||||||||||||||||||||||||||||
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Description
Talabostat is a non-selective inhibitor of dipeptidyl peptidases (DPPs), including DPP-4, DPP-7, DPP-8, DPP-9, fibroblast activation protein (FAP), and prolyl endopeptidase (PREP; IC50s = >4, 310, 4, 11, 560, and 390 nM, respectively). It inhibits proliferation of superantigen-stimulated human peripheral blood mononuclear cells (PBMCs; IC50 = ~10 nM). Talabostat (5 μg twice per day) increases expression of a variety of cytokines, including those encoding IL-1β, IL-6, and G-CSF, and chemokines in tumors and tumor-draining lymph nodes in a WEHI-164 fibrosarcoma mouse model. It reduces tumor growth in WEHI-164, MM45T.Sp, and MM52.T fibrosarcoma, EL-4 and A20/2J lymphoma, B16/F10 melanoma, and P815 mastocytoma syngeneic mouse models. Talabostat also increases the efficacy of the antitumor antibodies rituximab and trastuzumab in Namalwa B cell lymphoma and LS180 colon carcinoma mouse xenograft models, respectively.Related product price
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![[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate](https://img.chemicalbook.com/ProductImageEN/2019-12/small/ab6cf7f8-e28f-44c5-9373-aaa3f286bf0d.jpg){kind=small}
![[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate](/ProductImageEN/2022-08/small/2c7d7b32-26c1-41c0-ab6e-52984d69cdec.jpg){kind=small}