Paliperidone
|
- $5 - $9000
- Product name: Paliperidone
- CAS: 144598-75-4
- MF: C23H27FN4O3
- MW: 426.48
- EINECS:620-493-1
- MDL Number:MFCD00871802
- Synonyms:3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-Methyl-;Risperidone EP IMpurity C;Paliperidone 9-Hydroxyrisperidone;9-Hydroxyrisperidone solution;Risperidone Impurity 3(Risperidone EP Impurity C);Racemic Paliperidone;Paliperidone (9-Hydroxy Risperidone, Risperidone EP Impurity C);Paliperidone, 99%, a potent D2 and 5-HT2A antagonist
78 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- Ambeed
- ApexBio Technology
- Arctom
- AvaChem
- Biosynth
- Cayman Chemical
- Chemcia Scientific
- Chem-Impex
- ChemScene
- Chemtos
- Crysdot
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- Thermo Scientific Chemicals
- Tocris
- TRC
- Usbiological
Package
- 1mg
- 2.5mg
- 5mg
- 10mg
- 1ml of 1mg
- 25mg
- 50mg
- 100mg
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- 250mg
- 50
- 1mL
- 500mg
- 10
- 1g
- 1000mg
- 2000mg
- 2G
- 5g
- 5000mg
- 10g
- 25g
- 100000mg
- 1 g
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98%
- Packaging10mg
- Price$10
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98%
- Packaging50mg
- Price$14
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98%
- Packaging250mg
- Price$30
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98%
- Packaging1g
- Price$68
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98%
- Packaging5g
- Price$224
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98%
- Packaging25g
- Price$863
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product number10483
- Product descriptionPaliperidone 98%
- Packaging25G
- Price$640
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product number10483
- Product descriptionPaliperidone 98%
- Packaging5G
- Price$155
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberJ98586
- Product descriptionPaliperidone 95%
- Packaging1g
- Price$166
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ40100
- Product descriptionPaliperidone 98%(HPLC),powder
- Packaging50mg
- Price$101
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging50mg
- Price$116
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging25mg
- Price$62
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging5mg
- Price$41
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging1g
- Price$642
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberS451
- Product descriptionPaliperidone 98%(HPLC)
- Packaging5g
- Price$665
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ98586
- Product descriptionPaliperidone 95%
- Packaging5g
- Price$498
- Updated2026-06-04
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98% | 10mg | $10 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98% | 50mg | $14 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98% | 250mg | $30 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98% | 1g | $68 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98% | 5g | $224 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98% | 25g | $863 | 2026-05-28 | Buy |
| ACHEMBLOCK | 10483 | Paliperidone 98% | 25G | $640 | 2026-05-27 | Buy |
| ACHEMBLOCK | 10483 | Paliperidone 98% | 5G | $155 | 2026-05-27 | Buy |
| AK Scientific | J98586 | Paliperidone 95% | 1g | $166 | 2026-06-04 | Buy |
| AK Scientific | J40100 | Paliperidone 98%(HPLC),powder | 50mg | $101 | 2026-06-04 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 50mg | $116 | 2026-06-04 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 25mg | $62 | 2026-06-04 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 5mg | $41 | 2026-06-04 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 1g | $642 | 2026-06-04 | Buy |
| AK Scientific | S451 | Paliperidone 98%(HPLC) | 5g | $665 | 2026-06-04 | Buy |
| AK Scientific | J98586 | Paliperidone 95% | 5g | $498 | 2026-06-04 | Buy |
Properties
Melting point :158-160°C
Boiling point :612.3±65.0 °C(Predicted)
Density :1.45±0.1 g/cm3(Predicted)
Flash point :9℃
storage temp. :2-8°C
solubility :DMSO: soluble2mg/mL, clear (warmed)
pka :13.00±0.60(Predicted)
form :powder
color :white to brown
Henry's Law Constant :1.2×1015 mol/(m3Pa) at 25℃, HSDB (2015)
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.
InChI :InChI=1S/C23H27FN4O3/c1-14-17(23(30)28-9-2-3-19(29)22(28)25-14)8-12-27-10-6-15(7-11-27)21-18-5-4-16(24)13-20(18)31-26-21/h4-5,13,15,19,29H,2-3,6-12H2,1H3
InChIKey :PMXMIIMHBWHSKN-UHFFFAOYSA-N
SMILES :C12C(O)CCCN1C(=O)C(CCN1CCC(C3C4=C(ON=3)C=C(F)C=C4)CC1)=C(C)N=2
CAS DataBase Reference :144598-75-4(CAS DataBase Reference)
Boiling point :612.3±65.0 °C(Predicted)
Density :1.45±0.1 g/cm3(Predicted)
Flash point :9℃
storage temp. :2-8°C
solubility :DMSO: soluble2mg/mL, clear (warmed)
pka :13.00±0.60(Predicted)
form :powder
color :white to brown
Henry's Law Constant :1.2×1015 mol/(m3Pa) at 25℃, HSDB (2015)
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.
InChI :InChI=1S/C23H27FN4O3/c1-14-17(23(30)28-9-2-3-19(29)22(28)25-14)8-12-27-10-6-15(7-11-27)21-18-5-4-16(24)13-20(18)31-26-21/h4-5,13,15,19,29H,2-3,6-12H2,1H3
InChIKey :PMXMIIMHBWHSKN-UHFFFAOYSA-N
SMILES :C12C(O)CCCN1C(=O)C(CCN1CCC(C3C4=C(ON=3)C=C(F)C=C4)CC1)=C(C)N=2
CAS DataBase Reference :144598-75-4(CAS DataBase Reference)
Safety Information
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| Signal word: | Danger | ||||||||||||||
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Description
Paliperidone is a potent antagonist of dopamine receptors (IC50s = 1.0 and 0.9 nM for D2 and D3, respectively). It also avidly binds α1- and α2-adrenergic receptors, histamine H1 receptor, and serotonin (5-HT) receptors 5-HT1D and 5-HT2A (Kis = 10, 80, 3.4, 19, 1.2 nM, respectively). Paliperidone is also known as 9-hydroxy risperidone and is the major metabolite of the antipsychotic medication risperidone .Related product price
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Suppliers and manufacturers
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Shaanxi Dideu Medichem Co. Ltd
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CONIER CHEM AND PHARMA LIMITED
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