U 75875

U 75875 Suppliers list
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U 75875 Basic information
Product Name:U 75875
Synonyms:U 75875;N-(1-Naphtyloxyacetyl)-L-His-[(2R,3R,4R,5S)-3,4-dihydroxy-2-isopropyl-5-(cyclohexylmethyl)-5-amino*pentanoyl]-L-Ile-(2-pyridylmethyl)NH2;PNU-75875;(2R,3R,4R,5S)-6-cyclohexyl-3,4-dihydroxy-5-[[(2S)-3-(1H-imidazol-5-yl)-2-[(2-naphthalen-1-yloxyacetyl)amino]propanoyl]amino]-N-[(2S,3S)-3-methyl-1-oxo-1-(pyridin-2-ylmethylamino)pentan-2-yl]-2-propan-2-ylhexanamide;L-Idonamide, 6-cyclohexyl-2,5,6-trideoxy-5-[[(2S)-3-(1H-imidazol-4-yl)-2-[[(1-naphthalenyloxy)acetyl]amino]-1-oxopropyl]amino]-2-(1-methylethyl)-N-[(1S,2S)-2-methyl-1-[[(2-pyridinylmethyl)amino]carbonyl]butyl]-
CAS:112190-24-6
MF:C45H61N7O7
MW:812.01
EINECS:
Product Categories:
Mol File:112190-24-6.mol
U 75875 Structure
U 75875 Chemical Properties
Boiling point 1158.5±65.0 °C(Predicted)
density 1+-.0.06 g/cm3(Predicted)
pka12.71±0.46(Predicted)
Safety Information
MSDS Information
U 75875 Usage And Synthesis
UsesU 75875, is a peptidomimetic inhibitor, that inhibits HIV-1 gag-pol protein. In human peripheral blood mononuclear cells and in a continuous cell line, U-75875 completely blocked HIV replication, so it can be used as therapeutic potential of protease inhibitors for treatment of HIV infection.
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