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| | N-Desmethyl Rilmazolam Basic information |
| Product Name: | N-Desmethyl Rilmazolam | | Synonyms: | N-Desmethyl Rilmazolam;4H-[1,2,4]Triazolo[1,5-a][1,4]benzodiazepine-2-carboxamide, 8-chloro-6-(2-chlorophenyl)-N-methyl- | | CAS: | 50330-93-3 | | MF: | C18H13Cl2N5O | | MW: | 386.24 | | EINECS: | | | Product Categories: | | | Mol File: | 50330-93-3.mol |  |
| | N-Desmethyl Rilmazolam Chemical Properties |
| density | 1.527±0.14 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted) | | solubility | Acetonitrile: Soluble
Chloroform: Soluble
Methanol: Soluble | | pka | 8.484±0.40(predicted) |
| | N-Desmethyl Rilmazolam Usage And Synthesis |
| Uses | N-desmethyl Rilmazolam, a triazolobenzodiazepine, serves as an analytical reference standard. N-desmethyl Rilmazolam is an active metabolite derived from rilmazafone (HY-106547). N-desmethyl Rilmazolam is designed for use in research and forensic settings [1]. | | References | [1] Kronstrand R, et al.Rilmazafone: A designer benzodiazepine pro-drug involved infatal intoxications. J Anal Toxicol. 2023 Sep 15;47(7):640-643. DOI:10.1093/jat/bkad041
[2] MASAFUMI FUJIMOTO. Detection and determination of active metabolites of 1-(2-o-chlorobenzoyl-4-chlorophenyl)-5-glycyl-aminomethyl-3-dimethylcarbamoyl-1H-1,2,4-triazole hydrochloride dihydrate, (450191-S), in rat tissues, using a radioreceptor assay for benzodiazepines[J]. Biochemical pharmacology, 1984, 33 10: Pages 1645-1651. DOI: 10.1016/0006-2952(84)90287-9 |
| | N-Desmethyl Rilmazolam Preparation Products And Raw materials |
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