(Rac)-IDO1-IN-5 manufacturers
- (Rac)-IDO1-IN-5
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- $82.00
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2026-04-21
- CAS:2166616-74-4
- Purity:
- Supply Ability: 10g
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| | (Rac)-IDO1-IN-5 Basic information |
| Product Name: | (Rac)-IDO1-IN-5 | | Synonyms: | (Rac)-IDO1-IN-5;(Rac)-IDO-1-IN-5,(Rac) IDO1 IN 5,(Rac)IDO1IN5;Benzamide, N-[1-[2,3-dihydro-1-[(tetrahydro-2H-pyran-4-yl)carbonyl]-1H-indol-5-yl]ethyl]-4-fluoro- | | CAS: | 2166616-74-4 | | MF: | C23H25FN2O3 | | MW: | 396.45 | | EINECS: | | | Product Categories: | | | Mol File: | 2166616-74-4.mol |  |
| | (Rac)-IDO1-IN-5 Chemical Properties |
| Boiling point | 665.5±55.0 °C(Predicted) | | density | 1.251±0.06 g/cm3(Predicted) | | storage temp. | Store at -20°C | | solubility | Soluble in DMSO | | pka | 13.93±0.46(Predicted) | | form | Solid | | color | White to off-white |
| | (Rac)-IDO1-IN-5 Usage And Synthesis |
| Description | (Rac)-IDO1-IN-5 is a racemate of IDO1-IN-5. IDO1-IN-5 is a potent, selective and brain penetrated inhibitor of Indoleamine 2,3-Dioxygenase 1 (IDO1) activity, binds to apo-IDO1 lacking heme rather than mature heme-bound IDO1[1]. | | Uses | (Rac)-LY-3381916 ((Rac)-IDO1-IN-5; Example 1) is a racemate of LY-3381916[1]. LY-3381916 is a potent, selective and brain penetrated inhibitor of Indoleamine 2,3-Dioxygenase 1 (IDO1) activity, binds to apo-IDO1 lacking heme rather than mature heme-bound IDO1[2]. | | References | [1]. Frank C. Dorsey, et al. Abstract 5245: Identification and characterization of the IDO1 inhibitor LY3381916. Cancer Research. 2018, 78(13). |
| | (Rac)-IDO1-IN-5 Preparation Products And Raw materials |
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