Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate

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Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate Basic information
Product Name:Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate
Synonyms:4-THIAZOLEACETIC ACID, 2-AMINO-ALPHA-(METHOXYIMINO)-, ETHYL ESTER;4-THIAZOLEACETIC ACID, 2-AMINO-ALPHA-(METHOXYIMINO)-, ETHYL ESTER, (AZ)-;ethyl (EZ)-(2-aminothiazol-4-yl)-α-methoxyiminoacetate;ETHYL-2-METHOXY-AMINO-2-(2-AMINO-THIAZOLE-4-YL) ACETATE;ETHYL (2E)-2-(2-AMINO-1,3-THIAZOL-4-YL)-2-METHOXYIMINO-ACETATE;ETHYL (Z)-2-(2-AMINO-4-THIAZOLYL)-2-METHOXYIMINOACETATE;ethyl 2-amino-alpha-(methoxyimino)thiazol-4-acetate;2-AMINO-ALPHA-(METHOXYIMINO)-4-THIAZOLEACETIC ACID ETHYL ESTER
CAS:60846-15-3
MF:C8H11N3O3S
MW:229.26
EINECS:2624705
Product Categories:
Mol File:60846-15-3.mol
Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate Structure
Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate Chemical Properties
Melting point 162-164 °C(lit.)
Boiling point 363.4±34.0 °C(Predicted)
density 1.41±0.1 g/cm3(Predicted)
pka2.57±0.10(Predicted)
Safety Information
Hazard Codes Xi
Risk Statements 36/37/38
Safety Statements 26-37/39
WGK Germany 3
MSDS Information
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ACROS English
SigmaAldrich English
Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate Usage And Synthesis
Chemical PropertiesWhite crystals. Melting point 162-164°C (155-160°C).
UsesEthyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate is an intermediates (side chains) of third-generation cephalosporins, such as cefmenoxime, ceftriaxone, ceftriaxone, and cefotaxime.
SynthesisEthyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate can be obtained by oximation, methylation, bromination and cyclization with ethyl acetoacetate.
Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate Preparation Products And Raw materials
Raw materialsEthyl acetoacetate
Tag:Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate(60846-15-3) Related Product Information
4-Thiazoleacetic acid, 2-amino-alpha-(hydroxyimino) Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate Methyl 2-amino-4-thiazoleacetate 2-[(2-Aminothiazol-4-yl)ethoxycarbonylmethyleneaminooxy]-2-methylpropionic acid tert-butyl ester tert-Butyl N-(3-amino-3-thioxopropyl)carbamate ETHYL 2-(2-AMINOTHIAZOLE-4-YL)-2-METHOXYIMINOACETATE,Ethyl 2-(2-aminothiazole-4-yl)-2-methoxyiminoacetate(ATE) EHATA Ethyl 2-amino-4-thiazoleacetate 2-Aminothiazole-4-acetic acid Acetone oxime 2-(1,3-thiazol-4-yl)acetic acid 2-(2-Aminothiazole-4-yl)-2-methoxyiminoacetic acid 2-Amino-4-methylthiazole Acetaldoxime