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| | 1H-Imidazole, 2-(3,4-dihydro-5-methoxy-1H-2-benzopyran-1-yl)-4,5-dihydro- Basic information |
| | 1H-Imidazole, 2-(3,4-dihydro-5-methoxy-1H-2-benzopyran-1-yl)-4,5-dihydro- Chemical Properties |
| Boiling point | 455.3±45.0 °C(Predicted) | | density | 1.30±0.1 g/cm3(Predicted) | | pka | 9.78±0.40(Predicted) |
| | 1H-Imidazole, 2-(3,4-dihydro-5-methoxy-1H-2-benzopyran-1-yl)-4,5-dihydro- Usage And Synthesis |
| Uses | Tasipimidine is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 for human α2A-adrenoceptors. Tasipimidine can be utilized in research related to situational anxiety and fear[1]. | | IC 50 | Alpha-2A adrenergic receptor | | References | [1] Lehtimki J, et al. Tasipimidine-the pharmacological profile of a novel orally active selective α2A-adrenoceptor agonist. Eur J Pharmacol. 2022 May 15;923:174949. DOI:10.1016/j.ejphar.2022.174949 |
| | 1H-Imidazole, 2-(3,4-dihydro-5-methoxy-1H-2-benzopyran-1-yl)-4,5-dihydro- Preparation Products And Raw materials |
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