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| | 2-(6-CHLORO-3-PYRIDINYL)-9-AZABICYCLO[4.2.1]NON-2-ENE FUMARATE Basic information |
| | 2-(6-CHLORO-3-PYRIDINYL)-9-AZABICYCLO[4.2.1]NON-2-ENE FUMARATE Chemical Properties |
| Boiling point | 378.1±37.0 °C(Predicted) | | density | 1.189±0.06 g/cm3(Predicted) | | storage temp. | Desiccate at +4°C | | form | Powder | | pka | 9.58±0.40(Predicted) | | Water Solubility | Soluble to 100 mM in water with gentle warming |
| | 2-(6-CHLORO-3-PYRIDINYL)-9-AZABICYCLO[4.2.1]NON-2-ENE FUMARATE Usage And Synthesis |
| Uses | UB 165 Fumarate is a novel presynaptic nicotinic acetylcholine receptor (nAChRs) agonist, which shows immediate potency. | | Biological Activity | Subtype-selective nicotinic agonist. Full agonist at α 3 β 2- and very weak partial agonist at α 4 β 2- containing nAChRs. K i values are 0.27, 20 (IC 50 ), 2790 and 990 nM for α 4 β 2, α 3, α 7 and α 1 β 1 δ ε respectively. |
| | 2-(6-CHLORO-3-PYRIDINYL)-9-AZABICYCLO[4.2.1]NON-2-ENE FUMARATE Preparation Products And Raw materials |
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