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| | S(-)-win 55 212-3 mesylate Basic information |
| Product Name: | S(-)-win 55 212-3 mesylate | | Synonyms: | [(3S)-2,3-DIHYDRO-5-METHYL-3-(4-MORPHOLINYLMETHYL)PYRROLO[1,2,3-DE]-1,4-BENZOXAZIN-6-YL]-1-NAPHTHALENYL-METHANONE MONOMETHANESULFONATE;WIN 55,212-3 MESYLATE;S(-)-[2,3-Dihydro-5-methyl-3-[(4-morpholinyl)methyl]pyrrolo[1,2,3-de]-1,4-benzoxazinyl]-(1-naphthalenyl)methanone mesylate salt;S(-)-WIN 55,212-3 mesylate salt;[(3S)-2,3-Dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanonemonomethanesulfonate;FSGCSTPOPBJYSX-BDQAORGHSA-N;Methanone, [(3S)-2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-, methanesulfonate (1:1);(?)-WIN 55,212-3 mesylate | | CAS: | 131543-25-4 | | MF: | C27H26N2O3.CH4O3S | | MW: | 522.61 | | EINECS: | | | Product Categories: | | | Mol File: | 131543-25-4.mol |  |
| | S(-)-win 55 212-3 mesylate Chemical Properties |
| storage temp. | Store at +4°C | | solubility | 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 2.4 mg/mL | | form | solid | | color | off-white |
| | S(-)-win 55 212-3 mesylate Usage And Synthesis |
| Uses | WIN 552,12-3 Mesylate is a high affinity cannabinoid agonist. | | Biological Activity | Novel, low potency CB 2 receptor silent antagonist and CB 1 receptor partial inverse agonist. Competitively antagonizes effects of CP 55,940 (pA 2 = 6.1) and SR 144528 (pEC 50 = 5.3) at CB 2 receptors and acts as a partial inverse agonist at CB 1 receptors (pIC 50 = 5.5). Displays modest activity at human melatonin MT 1 and muscarinic M 4 receptors, but is selective over several other GPCRs. |
| | S(-)-win 55 212-3 mesylate Preparation Products And Raw materials |
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