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| | AM2201 N-(4-hydroxypentyl) metabolite Basic information |
| Product Name: | AM2201 N-(4-hydroxypentyl) metabolite | | Synonyms: | AM2201 N-(4-hydroxypentyl) metabolite;[1-(5-fluoro-4-hydroxypentyl)indol-3-yl]-naphthalen-1-ylmethanone;(1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone;AM-2201 4-hydroxypentyl metabolite;AM-2201 4-hydroxypenty metabolite;Methanone, [1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl]-1-naphthalenyl- | | CAS: | 1427521-34-3 | | MF: | C24H22FNO2 | | MW: | 375.44 | | EINECS: | | | Product Categories: | | | Mol File: | 1427521-34-3.mol |  |
| | AM2201 N-(4-hydroxypentyl) metabolite Chemical Properties |
| Boiling point | 603.6±50.0 °C(Predicted) | | density | 1.19±0.1 g/cm3(Predicted) | | solubility | Dichloromethane: 20 mg/ml; DMF: 20 mg/ml; DMSO: 20 mg/ml; Ethanol: 5 mg/ml | | pka | 13.87±0.20(Predicted) |
| | AM2201 N-(4-hydroxypentyl) metabolite Usage And Synthesis |
| Description | AM2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.1 AM2201 N-(4-hydroxypentyl) metabolite is an expected urinary metabolite of AM2201, based on the known metabolism of similar compounds.2 Its biological actions are unknown. | | Uses | 4-Hydroxypentyl AM-2201 is a metabolite of AM-2201 (A575830), is a drug which acts as a potent but unselective agonist for the cannabinoid receptor CB1 or CB2. | | References | 1. Makriyannis, A., and Deng, H. Cannabimimetic indole derivatives US7241799B2,(2001).
2. Wintermeyer, A., Mller, I., Thevis, M., et al. In vitro phase I metabolism of the synthetic cannabimimetic JWH-018 Anal. Bioanal. Chem. 398(5),2141-2153(2010). |
| | AM2201 N-(4-hydroxypentyl) metabolite Preparation Products And Raw materials |
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