| Company Name: |
BOC Sciences |
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1-631-485-4226; 16314854226 |
| Email: |
info@bocsci.com |
GSK299115A manufacturers
- GSK299115A
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- $336.00
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2026-07-14
- CAS:864082-35-9
- Purity: 99.87%
- Supply Ability: 10g
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| | GSK299115A Basic information |
| Product Name: | GSK299115A | | Synonyms: | GSK299115A;3-Pyridinecarboxamide, 4-(3,4-dichlorophenyl)-1,4,5,6-tetrahydro-N-1H-indazol-5-yl-2-methyl-6-oxo-;GSK299115A, 10 mM in DMSO | | CAS: | 864082-35-9 | | MF: | C20H16Cl2N4O2 | | MW: | 415.27 | | EINECS: | | | Product Categories: | | | Mol File: | 864082-35-9.mol |  |
| | GSK299115A Chemical Properties |
| Boiling point | 739.3±60.0 °C(Predicted) | | density | 1.479±0.06 g/cm3(Predicted) | | pka | 12.73±0.40(Predicted) |
| | GSK299115A Usage And Synthesis |
| Description | GSK299115A is a G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor (GRK2 inhibitor). G-protein-coupled receptor kinase 2 (GRK2) is a G-protein-coupled receptor kinase that is ubiquitously expressed in many tissues and regulates various intracellular mechanisms. GRK2 plays an important role in the maintenance of heart structure and function; thus, this kinase is involved in many cardiovascular diseases. | | Uses | GSK299115A is a G Protein-coupled Receptor Kinase (GRK) and PKA inhibitor[1]. | | References | [1] Homan KT, et al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10(1):310-9. DOI:10.1021/cb5006323 |
| | GSK299115A Preparation Products And Raw materials |
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