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Dasatinib N-Oxide

Dasatinib N-Oxide Suppliers list
Company Name: J & K SCIENTIFIC LTD.  
Tel: 18210857532 18210857532
Email: jkinfo@jkchemical.com
Company Name: Chemsky(shanghai)International Co.,Ltd.  
Tel: 021-50135380
Email: shchemsky@sina.com
Company Name: Daicel Chiral Technologies (China)CO.,LTD  
Tel: 021-50460086-9 15921403865
Email: han_yajun@dctc.daicel.com
Company Name: S.Z. PhyStandard Bio-Tech. Co., Ltd.  
Tel: 0755-83725681-603
Email:
Company Name: Clearsynth Labs Limited  
Tel: +91-22-26355700
Email: info@clearsynth.com

Dasatinib N-Oxide manufacturers

Dasatinib N-Oxide Basic information
Product Name:Dasatinib N-Oxide
Synonyms:Dasatinib N-Oxide;N-[2-Chloro-6-methylphenyl]-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamide N-Oxide;4-(6-((5-((2-chloro-6-methylphenyl)carbamoyl);N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-4-oxidopiperazin-4-ium-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide;Dasatinib impurity 4/Dasatinib N-Oxide/N-[2-Chloro-6-methylphenyl]-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamide N-Oxide;Dasatinib N4-Oxide;5-Thiazolecarboxamide, N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-4-oxido-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-;Dasatinib monohydrate A
CAS:910297-52-8
MF:C22H26ClN7O3S
MW:504.01
EINECS:
Product Categories:Intermediates & Fine Chemicals;Metabolites & Impurities;Pharmaceuticals;Sulfur & Selenium Compounds
Mol File:910297-52-8.mol
Dasatinib N-Oxide Structure
Dasatinib N-Oxide Chemical Properties
Melting point 193-195°C
storage temp. -20°C Freezer
solubility Acetonitrile (Slightly), DMSO (Slightly), Methanol (Slightly)
pka10.93±0.70(Predicted)
form Solid
color Off-White to Pale Yellow
Safety Information
HS Code 29349990
MSDS Information
Dasatinib N-Oxide Usage And Synthesis
Chemical PropertiesPale Yellow Solid
UsesAn oxidative metabolite of Dasatinib (M5 metabolite). It is a COVID19-related research product.
DefinitionChEBI: Dasatinib n-oxide is an aromatic amide.
in vivo

Dasatinib N-oxide is the pharmacologically active metabolite after oral administration[1].

Dasatinib N-Oxide Preparation Products And Raw materials
Tag:Dasatinib N-Oxide(910297-52-8) Related Product Information
Imatinib Sunitinib 5-Thiazolecarboxylic acid,2-[(6-chloro-2-Methyl-4-pyriMidinyl)aMino]- Des-6-[4-(2-hydroxyethyl)-1-piperazinyl]-6-chloro-O-pivalate Dasatinib Dasatinib DiMeric IMpurity Ibrutinib Dasatinib