SDZ SER 082 FUMARATE manufacturers
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| | SDZ SER 082 FUMARATE Basic information |
| Product Name: | SDZ SER 082 FUMARATE | | Synonyms: | SDZ SER 082 FUMARATE;(+)-CIS-4,5,7A,8,9,10,11,11A-OCTAHYDRO-7H-10-METHYLINDOLO[1,7-BC][2,6]-NAPHTHYRIDINE FUMARATE;SDZ SER 082;YASBOGFWAMXINH-TZMCWYRMSA-N;7H-Indolo[1,7-bc][2,6]naphthyridine, 4,5,7a,8,9,10,11,11a-octahydro-10-methyl-, (7aR,11aS)-rel- | | CAS: | 141474-54-6 | | MF: | C15H20N2 | | MW: | 228.33 | | EINECS: | | | Product Categories: | Serotonin receptor | | Mol File: | 141474-54-6.mol |  |
| | SDZ SER 082 FUMARATE Chemical Properties |
| Boiling point | 345.271±41.00 °C(Press: 760.00 Torr)(predicted) | | density | 1.172±0.10 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted) | | storage temp. | Store at RT | | pka | 9.795±0.20(predicted) | | Water Solubility | Soluble to 100 mM in Water |
| | SDZ SER 082 FUMARATE Usage And Synthesis |
| Uses | SDZ SER 082 is a 5-HT2C and 5-HT2B receptor antagonist. | | Uses | SDZ SER 082 Fumarate is a serotonin 2C receptor antagonist. | | Biological Activity | Selective 5-HT 2B/2C receptor antagonist with low affinity for 5-HT 1A receptors. Inhibits [ 3 H]-mesulergine binding to 5-HT 2C receptors with a pK D of 7.8. Inhibits 5-HT 2B mediated responses in the rat fundus (pK B = 7.34). |
| | SDZ SER 082 FUMARATE Preparation Products And Raw materials |
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