2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde

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2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde Basic information
Product Name:2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde
Synonyms:2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde;1H-Isoindole-5-carboxaldehyde, 2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-;2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbaldehyde;2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carbaldehyde;2-(2,6-Dioxo-3-piperidyl)-1,3-dioxoisoindoline-5-carbaldehyde;Thalidomide-5-carbaldehyde;2-(2,6-Dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindole-5-carboxaldehyde
CAS:1447701-63-4
MF:C14H10N2O5
MW:286.24
EINECS:
Product Categories:
Mol File:1447701-63-4.mol
2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde Structure
2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde Chemical Properties
Boiling point 584.9±45.0 °C(Predicted)
density 1.560±0.06 g/cm3(Predicted)
pka10.57±0.40(Predicted)
Safety Information
MSDS Information
2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde Usage And Synthesis
UsesThalidomide-5-carbaldehyde is a Thalidomide analogue with an aldehyde. Thalidomide recruiits E3 ligase for the ubiquitinylation and subsequent proteolysis of target proteins. The aldehyde is highly reactive towards amine nucleophiles through reductive amination among other reactions.
2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde Preparation Products And Raw materials
Tag:2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindoline-5-carbaldehyde(1447701-63-4) Related Product Information
Thalidomide CC-885 2-(2,6-dioxopiperidin-3-yl)-5-hydroxyisoindoline-1,3-dione 2-(2,6-dioxopiperidin-3-yl)-5-morpholinoisoindoline-1,3-dione (2S,4R)-1-((S)-2-amino-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide L-Prolinamide, 3-methyl-L-valyl-4-hydroxy-N-[(1S)-1-[4-(4-methyl-5-thiazolyl)phenyl]ethyl]-, (4R)-