beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2

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beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 Suppliers list
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beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 Basic information
Product Name:beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2
Synonyms:(B-MERCAPTO-B,B-CYCLOPENTAMETHYLENE-*PRO PIONYL1,O-E;[β-mercapto-β,β-cyclopentamethylenepropionyl1, o-et-tyr2, val4, arg8]-vasopressin;1-(1-MERCAPTOCYCLOHEXANEACETIC ACID)-2-(O-ETHYL-L-TYROSINE)-4-L- VALINE-8-L-ARGININEVASOPRESSIN;vasopressin 1-(1-MCHA)-2-(O-ethyl-L-tyrosine)-4-L-valine;[BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENEPROPIONYL1,O-ET-TYR2,VAL4,ARG8]-VASOPRESSIN;(D(CH2)(5/1),TYR(ET)2,VAL4,ARG8)-VASOPRESSIN;[1-MERCAPTOCYCLOHEXYL]ACETYL-TYR[O-ETHYL]-PHE-VAL-ASN-CYS-PRO-ARG-GLY-NH2;M.W. 1136.41 C53H77N13O11S2
CAS:77453-01-1
MF:C53H77N13O11S2
MW:1136.39
EINECS:
Product Categories:Vasopressin and Oxytocin receptor;Hormones;Oxytocin&Vasopressin;Pituitary Hormones;VasopressinPeptides for Cell Biology;Vasopressins
Mol File:77453-01-1.mol
beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 Structure
beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 Chemical Properties
storage temp. −20°C
form Solid
color White to off-white
Sequence{(1-Mercaptocyclohexyl)acetyl}-{Tyr(O-Ethyl)}-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge: 1-Cys6)
Safety Information
Hazard Codes Xn
Risk Statements 20
Safety Statements 36
WGK Germany 3
MSDS Information
ProviderLanguage
SigmaAldrich English
beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 Usage And Synthesis
UsesSKF 100398 (d(CH2)5Tyr(Et)VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP[1].
in vivo

SKF 100398 is a specific antagonist of the hydrosmotic effect of exogenous and endogenous AVP[1].
SKF 100398 (8 μg/kg; i.v.) abolishes the antidiuretic effect of AVP[1].

Animal Model:Male Sprague-Dawley rats (250-300 g)[1]
Dosage:8 μg/kg
Administration:Intravenous injection
Result:Completely blocked the antidiuretic effect of exogenous AVP (4 ng/kg body wt i.v.).
References[1] S Ishikawa, et al. Further in vivo evidence for antagonist-to-antidiuretic action of arginine vasopressin. Am J Physiol. 1983 Nov;245(5 Pt 1):R713-9. DOI:10.1152/ajpregu.1983.245.5.R713
beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2 Preparation Products And Raw materials
Raw materialsGlycinamide, O-ethyl-N-[(1-mercaptocyclohexyl)acetyl]-D-tyrosyl-L-phenylalanyl-L-valyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-arginyl- (9CI)
Tag:beta-Mercapto-beta,beta-cyclopentamethylene-propionyl-Tyr(Et)-Phe-Val-Asn-Cys-Pro-Arg-Gly-NH2(77453-01-1) Related Product Information
2-Methyl-2-pentanethiol 3-(4-Methoxyphenyl)propionamide N-Octyl-ethylene-1,2-diamine METHYL PENTYL DISULPHIDE BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-TYR(ET)-PHE-VAL-ASN-CYS-PRO-ARG-NH2 BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-TYR(ET)-PHE-VAL-ASN-CYS-PRO-ARG-GLY-NH2 isopropyl propyl disulphide 3-ETHYL-3-PENTANETHIOL Cyclohexyl mercaptan N-(4-Methoxyphenethyl)acetamide