中文名:酪氨酸激酶抑制剂AG 490
英文名:AG-490 (Tyrphostin B42)
应用:Tyrphostin AG has been used to block IL-6 cytokine signaling to study its effects on glial cell reactivity. AG 490 has also been used as a JAK2 inhibitor in human umbilical vein endothelial cells
纯度:Moligand™,≥98%
货号:A126525
Cas号:133550-30-8
存储温度:-20°C储存
运输条件:超低温运输
产品介绍:
AG-490 (Tyrphostin AG 490)是EGFR抑制剂,IC50为100nM,比对ErbB2的抑制性高135倍,对Lck,Lyn,Btk,Syk和Src无活性。Tyrphostin AG has been used to block IL-6 cytokine signaling to study its effects on glial cell reactivity. AG 490 has also been used as a JAK2 inhibitor in human umbilical vein endothelial cells
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