ARV-771
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- $13 - $4173.5
- Product name: ARV-771
- CAS: 1949837-12-0
- MF: C49H60ClN9O7S2
- MW: 986.65
- EINECS:
- MDL Number:MFCD30738017
- Synonyms:ARV-771;ARV 771; ARV771;(2S,4R)-1-[(2S)-2-[[2-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide;(2S,4R)-1-[(2S)-2-[[2-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-;(2S,4R)-1-((2S)-2-(tert-butyl)-15-((6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,14-dioxo-6,10-dioxa-3,13-diazapentadecan-1-oyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide;Epigenetic Reader Domain,ARV-771,ARV771,inhibit,ARV 771,PROTACs,Inhibitor;ARV-771, 10 mM in DMSO;(2S,4R)-1-[(S)-2-(tert-Butyl)-15-[(S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-4,14-dioxo-6,10-dioxa-3,13-diazapentadecan-1-oyl]-4-hydroxy-N-[(S)-1-[4-(4-methyl-5-thiazolyl)phenyl]ethyl]pyrrolidine-2-carboxamide
50 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- ApexBio Technology
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- Chemenu
- ChemScene
- DC Chemicals
- Matrix Scientific
- Tocris
Package
- 5
- 1mg
- 5mg
- 10.00mg
- 10mg
- 25.00mg
- 25mg
- 50.00mg
- 50mg
- 100mg
- 200mg
- 250mg
- 1mL(10mMinDMSO)
- 1g
- 10mM*1mLinDMSO
- 1mlx10mM(inDMSO)
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 ≥98%
- Packaging1mg
- Price$13
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 ≥98%
- Packaging5mg
- Price$48
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 98%
- Packaging10mg
- Price$63
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 97%
- Packaging25mg
- Price$128
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 97%
- Packaging50mg
- Price$253
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 97%
- Packaging100mg
- Price$431
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 96%
- Packaging250mg
- Price$798
- Updated2026-05-30
- Buy
- Manufactureraablocks
- Product numberAA01EO2W
- Product descriptionARV-771 96%
- Packaging1g
- Price$2356
- Updated2026-05-30
- Buy
- ManufacturerACHEMBLOCK
- Product numberK16213
- Product descriptionARV-771 98%
- Packaging100MG
- Price$510
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberK16213
- Product descriptionARV-771 98%
- Packaging25MG
- Price$175
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product number2258EJ
- Product description(2S,4R)-1-[(2S)-2-[[2-[3-[2-[[2-[(9S)-7-(4-Chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide
- Packaging10mg
- Price$768
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberBA4656
- Product descriptionARV-771
- Packaging1mL(10mMinDMSO)
- Price$234
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA4656
- Product descriptionARV-771
- Packaging10mg
- Price$216
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA4656
- Product descriptionARV-771
- Packaging5mg
- Price$135
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA4656
- Product descriptionARV-771
- Packaging1mg
- Price$63
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA4656
- Product descriptionARV-771
- Packaging50mg
- Price$801
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA01EO2W | ARV-771 ≥98% | 1mg | $13 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 ≥98% | 5mg | $48 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 98% | 10mg | $63 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 97% | 25mg | $128 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 97% | 50mg | $253 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 97% | 100mg | $431 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 96% | 250mg | $798 | 2026-05-30 | Buy |
| aablocks | AA01EO2W | ARV-771 96% | 1g | $2356 | 2026-05-30 | Buy |
| ACHEMBLOCK | K16213 | ARV-771 98% | 100MG | $510 | 2026-05-27 | Buy |
| ACHEMBLOCK | K16213 | ARV-771 98% | 25MG | $175 | 2026-05-27 | Buy |
| AK Scientific | 2258EJ | (2S,4R)-1-[(2S)-2-[[2-[3-[2-[[2-[(9S)-7-(4-Chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide | 10mg | $768 | 2021-12-16 | Buy |
| ApexBio Technology | BA4656 | ARV-771 | 1mL(10mMinDMSO) | $234 | 2026-05-06 | Buy |
| ApexBio Technology | BA4656 | ARV-771 | 10mg | $216 | 2026-05-06 | Buy |
| ApexBio Technology | BA4656 | ARV-771 | 5mg | $135 | 2026-05-06 | Buy |
| ApexBio Technology | BA4656 | ARV-771 | 1mg | $63 | 2026-05-06 | Buy |
| ApexBio Technology | BA4656 | ARV-771 | 50mg | $801 | 2026-05-06 | Buy |
Properties
Density :1.39±0.1 g/cm3(Predicted)
storage temp. :Sealed in dry,Store in freezer, under -20°C
solubility :DMSO:65.92(Max Conc. mg/mL);68.22(Max Conc. mM)
DMF:20.0(Max Conc. mg/mL);20.7(Max Conc. mM)
DMF:PBS (pH 7.2) (1:6):0.14(Max Conc. mg/mL);0.14(Max Conc. mM)
Ethanol:55.0(Max Conc. mg/mL);56.92(Max Conc. mM) form :A crystalline solid
pka :13.61±0.46(Predicted)
color :White to light yellow
InChIKey :PQOGZKGXGLHDGS-BZTQNJCZNA-N
SMILES :[s]1cnc(c1c2ccc(cc2)[C@@H](NC(=O)[C@H]3N(C[C@@H](C3)O)C(=O)[C@@H](NC(=O)COCCCOCCNC(=O)C[C@@H]4N=C(c6c([s]c(c6C)C)[n]7c4nnc7C)c5ccc(cc5)Cl)C(C)(C)C)C)C
storage temp. :Sealed in dry,Store in freezer, under -20°C
solubility :DMSO:65.92(Max Conc. mg/mL);68.22(Max Conc. mM)
DMF:20.0(Max Conc. mg/mL);20.7(Max Conc. mM)
DMF:PBS (pH 7.2) (1:6):0.14(Max Conc. mg/mL);0.14(Max Conc. mM)
Ethanol:55.0(Max Conc. mg/mL);56.92(Max Conc. mM) form :A crystalline solid
pka :13.61±0.46(Predicted)
color :White to light yellow
InChIKey :PQOGZKGXGLHDGS-BZTQNJCZNA-N
SMILES :[s]1cnc(c1c2ccc(cc2)[C@@H](NC(=O)[C@H]3N(C[C@@H](C3)O)C(=O)[C@@H](NC(=O)COCCCOCCNC(=O)C[C@@H]4N=C(c6c([s]c(c6C)C)[n]7c4nnc7C)c5ccc(cc5)Cl)C(C)(C)C)C)C
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||||||||||||||||
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| Precautionary statements: |
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Description
ARV-771 is a BET PROTAC based on E3 ligase von Hippel-Lindau with Kds of 34 nM, 4.7 nM, 8.3 nM, 7.6 nM, 9.6 nM, and 7.6 nM for BRD2(1), BRD2(2), BRD3(1), BRD3(2), BRD4(1) and BRD4(2), respectively.Suppliers and manufacturers
Wuhan Fortuna Chemical Co., Ltd
BOC Sciences
Zhengzhou Alfa Chemical Co.,Ltd
Career Henan Chemica Co
Zhejiang J&C Biological Technology Co.,Limited
HANGZHOU LEAP CHEM CO., LTD.
TargetMol Chemicals Inc.
Zibo Hangyu Biotechnology Development Co., Ltd
Shanghai Acmec Biochemical Technology Co., Ltd.
ARV-771
CAS:1949837-12-0