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ChemicalBook >> CAS DataBase List >> Sitravatinib

Sitravatinib

Sitravatinib price.
  • $22 - $1600
  • Product name: Sitravatinib
  • CAS: 1123837-84-2
  • MF: C33H29F2N5O4S
  • MW: 629.68
  • EINECS:
  • MDL Number:MFCD28502181
  • Synonyms:CS-2638;Sitravatinib;N-(3-fluoro-4-((2-(5-(((2-methoxyethyl)amino)methyl)pyridin-2-yl)thieno[3,2-b]pyridin-7-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide;MGCD-516;MG516;Sitravatinib (MGCD516);1,1-Cyclopropanedicarboxamide, N-[3-fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-;RTK,MG-516,PD-1,SCFR,DDR1,inhibit,VEGFR2,MG 516,MGCD 516,MER,immune,TRKA,Cluster of differentiation antigen 135,Cancer,Discoidin Domain Receptor,VEGFR3,Inhibitor,Vascular endothelial growth factor receptor,Trk Receptor,Tropomyosin related kinase receptor,CD135,VEGFR,immunotherapy,Macrophages,c-Kit,DDR2,VEGFR1,Tyrosine,Fms like tyrosine kinase 3,FLT3,Axl,TRKB,Sitravatinib,MGCD-516,KIT,kinase,CD117
Price51 Properties Safety Information Description
51 prices
Selected condition：
Brand
  • aablocks
  • ACHEMBLOCK
  • AK Scientific
  • ApexBio Technology
  • Arctom
  • AvaChem
  • Biosynth
  • Cayman Chemical
  • ChemScene
  • Crysdot
  • DC Chemicals
  • TRC
  • Usbiological
Package
  • 10mM(1mLinDMSO)
  • 10mM*1mLinDMSO(Solution)
  • 10mM*1mLinDMSO(Solid+Solvent)
  • 10mM*1mLinDMSO
  • 1mg
  • 5mg
  • 10mg
  • 20mg
  • 25mg
  • 50mg
  • 100mg
  • 200mg
  • 250mg
  • 500mg
  • 1g
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98%
  • Packaging1mg
  • Price$22
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98%
  • Packaging5mg
  • Price$35
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98%
  • Packaging10mg
  • Price$52
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98%
  • Packaging25mg
  • Price$98
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98%
  • Packaging50mg
  • Price$157
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98%
  • Packaging100mg
  • Price$250
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98
  • Packaging200mg
  • Price$471
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA008TMR
  • Product descriptionN-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98
  • Packaging500mg
  • Price$732
  • Updated2026-05-28
  • Buy
  • ManufacturerACHEMBLOCK
  • Product numberY228285
  • Product descriptionSitravatinib 97.00%
  • Packaging100MG
  • Price$425
  • Updated2026-05-27
  • Buy
  • ManufacturerACHEMBLOCK
  • Product numberY228285
  • Product descriptionSitravatinib 97.00%
  • Packaging25MG
  • Price$165
  • Updated2026-05-27
  • Buy
  • ManufacturerAK Scientific
  • Product number3193DC
  • Product descriptionSitravatinib
  • Packaging5mg
  • Price$151
  • Updated2021-12-16
  • Buy
  • ManufacturerAK Scientific
  • Product number3193DC
  • Product descriptionSitravatinib
  • Packaging10mg
  • Price$205
  • Updated2021-12-16
  • Buy
  • ManufacturerApexBio Technology
  • Product numberA4695
  • Product descriptionSitravatinib
  • Packaging10mg
  • Price$100
  • Updated2026-05-06
  • Buy
  • ManufacturerApexBio Technology
  • Product numberA4695
  • Product descriptionSitravatinib
  • Packaging5mg
  • Price$64
  • Updated2026-05-06
  • Buy
  • ManufacturerArctom
  • Product numberSLK-S8573
  • Product descriptionSitravatinib (MGCD516) 99.97%
  • Packaging5mg
  • Price$140
  • Updated2026-05-26
  • Buy
  • ManufacturerArctom
  • Product numberHY-16961
  • Product descriptionSitravatinib 99.57%
  • Packaging5mg
  • Price$57
  • Updated2026-05-26
  • Buy
Manufacturer Product number Product description Packaging Price Updated Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98% 1mg $22 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98% 5mg $35 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98% 10mg $52 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98% 25mg $98 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98% 50mg $157 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98% 100mg $250 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98 200mg $471 2026-05-28 Buy
aablocks AA008TMR N-[3-Fluoro-4-[[2-[5-[[(2-methoxyethyl)amino]methyl]-2-pyridinyl]thieno[3,2-b]pyridin-7-yl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide 98 500mg $732 2026-05-28 Buy
ACHEMBLOCK Y228285 Sitravatinib 97.00% 100MG $425 2026-05-27 Buy
ACHEMBLOCK Y228285 Sitravatinib 97.00% 25MG $165 2026-05-27 Buy
AK Scientific 3193DC Sitravatinib 5mg $151 2021-12-16 Buy
AK Scientific 3193DC Sitravatinib 10mg $205 2021-12-16 Buy
ApexBio Technology A4695 Sitravatinib 10mg $100 2026-05-06 Buy
ApexBio Technology A4695 Sitravatinib 5mg $64 2026-05-06 Buy
Arctom SLK-S8573 Sitravatinib (MGCD516) 99.97% 5mg $140 2026-05-26 Buy
Arctom HY-16961 Sitravatinib 99.57% 5mg $57 2026-05-26 Buy
Next Last

Properties

Boiling point :833.5±65.0 °C(Predicted)
Density :1.417±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :Soluble in DMSO (up to at least 25 mg/ml), or in Ethanol (up to at least 25 mg/ml)
form :solid
pka :13.17±0.70(Predicted)
color :Off-white
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
InChIKey :WLAVZAAODLTUSW-UHFFFAOYSA-N
SMILES :C1(C(NC2=CC=C(F)C=C2)=O)(C(NC2=CC=C(OC3C=CN=C4C=C(C5=NC=C(CNCCOC)C=C5)SC4=3)C(F)=C2)=O)CC1

Safety Information

Symbol(GHS): Exclamation Mark (GHS07)
Signal word: Warning
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
H302 Harmful if swallowed Acute toxicity,oral Category 4 Warning P264, P270, P301+P312, P330, P501
H315 Causes skin irritation Skin corrosion/irritation Category 2 Warning P264, P280, P302+P352, P321,P332+P313, P362
H319 Causes serious eye irritation Serious eye damage/eye irritation Category 2A Warning P264, P280, P305+P351+P338,P337+P313P
H335 May cause respiratory irritation Specific target organ toxicity, single exposure;Respiratory tract irritation Category 3 Warning
Precautionary statements:
P261 Avoid breathing dust/fume/gas/mist/vapours/spray.
P305+P351+P338 IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

Description

Sitravatinib, known as MGCD516, is a multikinase (MET, RET, AXL, NTRK1, or NTRK3 genes) inhibitor used in a phase 1/1b clinical trial (NCT02219711) for patients with advanced cancers (NCT02219711).

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Suppliers and manufacturers

Suzhou Meidi Senuo Pharmaceutical Technology Co., Ltd. Dalian Meilun Biotech Co., Ltd. MedChemexpress LLC Bide Pharmatech Ltd. Shanghai Lollane Biological Technology Co.,Ltd. Shanghai YuanYe Biotechnology Co., Ltd. Qingdao IniKem BioPharmaTech Co.,Ltd ShangHai Biochempartner Co.,Ltd Shanghai Zhixin Chemical Technology Co., Ltd. Amadis Chemical Company Limited