| Identification | Back Directory | [Name]
Benzenepropanamide, α-[[(1,2-dihydro-2-oxo-6-quinolinyl)sulfonyl]amino]-N-(2-furanylmethyl)-N-(2-thienylmethyl)-, (αR)- | [CAS]
1681056-62-1 | [Synonyms]
PG 34
Benzenepropanamide, α-[[(1,2-dihydro-2-oxo-6-quinolinyl)sulfonyl]amino]-N-(2-furanylmethyl)-N-(2-thienylmethyl)-, (αR)- | [Molecular Formula]
C28H25N3O5S2 | [MOL File]
1681056-62-1.mol | [Molecular Weight]
547.64 |
| Hazard Information | Back Directory | [Uses]
PG 34 is a weak O-GlcNAc transferase (OGT) inhibitor (IC50=68 μM), and a close structural analog of OSMI-1.html" class="link-product" target="_blank">OSMI-1 (HY-119738)[1]. | [References]
[1] Rodrigo F Ortiz-Meoz, et al. A small molecule that inhibits OGT activity in cells. ACS Chem Biol. 2015 Jun 19;10(6):1392-7. DOI:10.1021/acschembio.5b00004 |
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