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Dersimelagon phosphate

Dersimelagon phosphate Structure
Dersimelagon phosphate structure
CAS No.
2490660-87-0
Chemical Name:
Dersimelagon phosphate
Synonyms
Dersimelagon phosphate
CBNumber:
CB013380476
Molecular Formula:
C36H45F4N3O5.H3O4P
Molecular Weight:
773.75
MDL Number:
MOL File:
2490660-87-0.mol
MSDS File:
SDS
Last updated:2025-04-18 09:51:25
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Dersimelagon phosphate Properties

FDA UNII 7GHY3N4EDN

Dersimelagon phosphate Chemical Properties, Uses, Production

Uses

Dersimelagon phosphate is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively. Dersimelagon phosphate shows good affinity for hMC1R and hMC4R with Ki values of 2.26, 32.9 nM, respectively. Dersimelagon phosphate can be used for the research of skin pigmentation[1][2].

References

[1] T. Suzuki, et al. Melanogenic effect of dersimelagon (MT-7117), a novel oral melanocortin 1 receptor agonist. Skin Health Dis. 2022; 2(1):e78.
[2] Erwin AL, et al. Porphyrias in the Age of Targeted Therapies. Diagnostics (Basel). 2021;11(10):1795. Published 2021 Sep 29. DOI:10.3390/diagnostics11101795

Dersimelagon phosphate Preparation Products And Raw materials

Raw materials

Preparation Products

Dersimelagon phosphate Suppliers

Global Suppliers ( 1)
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
Supplier Advantage
TargetMol Chemicals Inc. 58

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Dersimelagon phosphate 2490660-87-0