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BRD4 Inhibitor-28

BRD4 Inhibitor-28 Structure
BRD4 Inhibitor-28 structure
CAS No.
2468960-80-5
Chemical Name:
BRD4 Inhibitor-28
Synonyms
BRD4 Inhibitor-28;Imidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one, 8-(1,6-dihydro-1,5-dimethyl-6-oxo-3-pyridinyl)-4,5-dihydro-1-(phenylmethyl)-
CBNumber:
CB014133686
Molecular Formula:
C23H21N3O3
Molecular Weight:
387.43
MDL Number:
MOL File:
2468960-80-5.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-05-11 15:21:01
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BRD4 Inhibitor-28 Properties

Boiling point 630.533±55.00 °C(Press: 760.00 Torr)(predicted)
Density 1.397±0.10 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted)
pka 2.233±0.20(predicted)

BRD4 Inhibitor-28 Chemical Properties, Uses, Production

Uses

BRD4 Inhibitor-28 (Compound 18) is an orally active BRD4 Inhibitor. BRD4 Inhibitor-28 inhibits BRD40-BD1, BRD40-BD2 with IC50s of 15, 55 nM. BRD4 Inhibitor-28 also inhibits BRD2-BD1, BRD3-BD1, BRDT-BD1 with IC50s of 19, 25, 68 nM. BRD4 Inhibitor-28 has anti-melanoma activity[1].

References

[1] Horai Y, et al. Discovery of a potent, orally available tricyclic derivative as a novel BRD4 inhibitor for melanoma. Bioorg Med Chem. 2023 Aug 26;93:117461. DOI:10.1016/j.bmc.2023.117461

BRD4 Inhibitor-28 Preparation Products And Raw materials

Raw materials

Preparation Products

BRD4 Inhibitor-28 Suppliers

Global Suppliers ( 2)
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
TargetMol Chemicals Inc. 13564774135 marketing@targetmol.com United States 19950 58
Supplier Advantage
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58

View Latest Price from BRD4 Inhibitor-28 manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
BRD4 Inhibitor-28 pictures 2026-05-11 BRD4 Inhibitor-28
2468960-80-5
 $1670.00-2800.00 10g TargetMol Chemicals Inc.

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BRD4 Inhibitor-28 Imidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one, 8-(1,6-dihydro-1,5-dimethyl-6-oxo-3-pyridinyl)-4,5-dihydro-1-(phenylmethyl)- 2468960-80-5