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hTG2 inhibitor VA4 (VA4)

hTG2 inhibitor VA4 (VA4) Structure
hTG2 inhibitor VA4 (VA4) structure
CAS No.
2088001-23-2
Chemical Name:
hTG2 inhibitor VA4 (VA4)
Synonyms
VA4;VA4 TG2 inhibitor;hTG2 inhibitor VA4 (VA4);Benzyl(S)-(6-acrylamido-1-(4-((5-(dimethylamino)naphthalen-1-yl)sulfonyl)piperazin-1-yl)-1-oxohexan-2-yl)carbamate;Carbamic acid, N-[(1S)-1-[[4-[[5-(dimethylamino)-1-naphthalenyl]sulfonyl]-1-piperazinyl]carbonyl]-5-[(1-oxo-2-propen-1-yl)amino]pentyl]-, phenylmethyl ester
CBNumber:
CB24844879
Molecular Formula:
C33H41N5O6S
Molecular Weight:
635.77
MDL Number:
MOL File:
2088001-23-2.mol
MSDS File:
SDS
Last updated:2026-07-16 07:06:08
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hTG2 inhibitor VA4 (VA4) Properties

Density 1.266±0.06 g/cm3(Predicted)
form Solid
pka 11.47±0.46(Predicted)
color Light yellow to yellow

hTG2 inhibitor VA4 (VA4) price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
ChemScene CS-0088463 TG2 inhibitor VA4 99.66% 2088001-23-2 5mg $146 2026-06-04 Buy
ChemScene CS-0088463 TG2 inhibitor VA4 99.66% 2088001-23-2 10mg $238 2026-06-04 Buy
ChemScene CS-0088463 TG2 inhibitor VA4 99.66% 2088001-23-2 25mg $471 2026-06-04 Buy
ChemScene CS-0088463 TG2 inhibitor VA4 99.66% 2088001-23-2 50mg $758 2026-06-04 Buy
aablocks AA0201BK Benzyl(S)-(6-acrylamido-1-(4-((5-(dimethylamino)naphthalen-1-yl)sulfonyl)piperazin-1-yl)-1-oxohexan-2-yl)carbamate 95%byHPLC 2088001-23-2 5mg $412 2026-06-01 Buy
Product number Packaging Price Buy
CS-0088463 5mg $146 Buy
CS-0088463 10mg $238 Buy
CS-0088463 25mg $471 Buy
CS-0088463 50mg $758 Buy
AA0201BK 5mg $412 Buy

hTG2 inhibitor VA4 (VA4) Chemical Properties,Uses,Production

Description

VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.

Uses

hTG2 inhibitor VA4 (compound VA4) is an irreversible Type 2 transglutaminase (TG2) inhibitor. hTG2 inhibitor VA4 reacts exclusively at the TG2 transamidase site, inhibits both transamidase and GTP-binding activities[1].

References

[1] Kerr C, et al. Transamidase site-targeted agents alter the conformation of the transglutaminase cancer stem cell survival protein to reduce GTP binding activity and cancer stem cell survival. Oncogene. 2017 May 25;36(21):2981-2990. DOI:10.1038/onc.2016.452

hTG2 inhibitor VA4 (VA4) Preparation Products And Raw materials

Raw materials

Preparation Products

hTG2 inhibitor VA4 (VA4) Suppliers

Global( 2)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
TargetMol Chemicals Inc. 13564774135 marketing@targetmol.com United States 19950 58
Supplier Advantage
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58

View Lastest Price from hTG2 inhibitor VA4 (VA4) manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
VA4 TG2 inhibitor pictures 2026-07-15 VA4 TG2 inhibitor
2088001-23-2
 $1520.00-2500.00 10g TargetMol Chemicals Inc.

2088001-23-2(hTG2 inhibitor VA4 (VA4))Related Search:

hTG2 inhibitor VA4 (VA4) 8,11-Dioxa-2,5-diazatridecanoic acid, 13-[[[5-(dimethylamino)-1-naphthalenyl]sulfonyl]amino]-4-oxo-3-[4-[(1-oxo-2-propen-1-yl)amino]butyl]-, phenylmethyl ester, (3S)- Benzamide, 3,4-dimethoxy-N-[5-[[4-[(1-oxo-2-propen-1-yl)amino]-1-piperidinyl]sulfonyl]-1-naphthalenyl]- ZED-1227 1,3-dimethyl-2-((2-oxopropyl)thio)imidazolium
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hTG2 inhibitor VA4 (VA4) VA4 Carbamic acid, N-[(1S)-1-[[4-[[5-(dimethylamino)-1-naphthalenyl]sulfonyl]-1-piperazinyl]carbonyl]-5-[(1-oxo-2-propen-1-yl)amino]pentyl]-, phenylmethyl ester Benzyl(S)-(6-acrylamido-1-(4-((5-(dimethylamino)naphthalen-1-yl)sulfonyl)piperazin-1-yl)-1-oxohexan-2-yl)carbamate VA4 TG2 inhibitor 2088001-23-2