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GSK299115A

CAS No.
864082-35-9
Chemical Name:
GSK299115A
Synonyms
GSK299115A;GSK299115A, 10 mM in DMSO;3-Pyridinecarboxamide, 4-(3,4-dichlorophenyl)-1,4,5,6-tetrahydro-N-1H-indazol-5-yl-2-methyl-6-oxo-
CBNumber:
CB54919749
Molecular Formula:
C20H16Cl2N4O2
Molecular Weight:
415.27
MDL Number:
MOL File:
864082-35-9.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-07-14 16:49:18

GSK299115A Properties

Boiling point 739.3±60.0 °C(Predicted)
Density 1.479±0.06 g/cm3(Predicted)
pka 12.73±0.40(Predicted)

GSK299115A price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
ChemScene CS-0082887 GSK299115A 98.99% 864082-35-9 1mg $619 2026-06-04 Buy
aablocks AA024C96 GSK299115A 864082-35-9 1mg $289 2026-06-01 Buy
aablocks AA024C96 GSK299115A 864082-35-9 5mg $671 2026-06-01 Buy
aablocks AA024C96 GSK299115A 864082-35-9 10mg $924 2026-06-01 Buy
aablocks AA024C96 GSK299115A 864082-35-9 25mg $1364 2026-06-01 Buy
Product number Packaging Price Buy
CS-0082887 1mg $619 Buy
AA024C96 1mg $289 Buy
AA024C96 5mg $671 Buy
AA024C96 10mg $924 Buy
AA024C96 25mg $1364 Buy

GSK299115A Chemical Properties, Uses, Production

Description

GSK299115A is a G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor (GRK2 inhibitor). G-protein-coupled receptor kinase 2 (GRK2) is a G-protein-coupled receptor kinase that is ubiquitously expressed in many tissues and regulates various intracellular mechanisms. GRK2 plays an important role in the maintenance of heart structure and function; thus, this kinase is involved in many cardiovascular diseases.

Uses

GSK299115A is a G Protein-coupled Receptor Kinase (GRK) and PKA inhibitor[1].

References

[1] Homan KT, et al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10(1):310-9. DOI:10.1021/cb5006323

GSK299115A Preparation Products And Raw materials

Raw materials

Preparation Products

GSK299115A Suppliers

Global Suppliers ( 10)
Supplier Tel Email Country ProdList Advantage
BOC Sciences 1-631-485-4226; 16314854226 info@bocsci.com United States 9920 65
TargetMol Chemicals Inc. +1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
Nantong QuanYi Biotechnology Co., Ltd 0513-66337626 18051384581 sales@chemhifuture.com China 5985 58
Shanghai Yifei Biotechnology Co. , Ltd. 021-65675885 18964387627 customer_service@efebio.com China 11963 58
RD International Technology Co., Limited 18024082417 market@ubiochem.com China 9831 58
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
Shanghai Amole Biotechnology Co., Ltd. 13370042665 18916960931 2596183085@qq.com China 17234 58

View Latest Price from GSK299115A manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
GSK299115A pictures 2026-07-14 GSK299115A
864082-35-9
$336.00-1130.00 99.87% 10g TargetMol Chemicals Inc.
  • GSK299115A pictures
  • GSK299115A
    864082-35-9
  • $336.00-1130.00
  • 99.87%
  • TargetMol Chemicals Inc.

GSK299115A Spectrum

GSK299115A 3-Pyridinecarboxamide, 4-(3,4-dichlorophenyl)-1,4,5,6-tetrahydro-N-1H-indazol-5-yl-2-methyl-6-oxo- GSK299115A, 10 mM in DMSO 864082-35-9