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c-Kit-IN-2

c-Kit-IN-2 Structure
c-Kit-IN-2 structure
CAS No.
2121515-37-3
Chemical Name:
c-Kit-IN-2
Synonyms
c-Kit-IN-2;c Kit IN 2,cKitIN2;Urea, N-(5-ethyl-3-isoxazolyl)-N'-[4-[2-[[6-(4-ethyl-1-piperazinyl)-4-pyrimidinyl]amino]-5-thiazolyl]phenyl]-
CBNumber:
CB58054341
Molecular Formula:
C25H29N9O2S
Molecular Weight:
519.62
MDL Number:
MFCD32067981
MOL File:
2121515-37-3.mol
MSDS File:
SDS
Last updated:2026-07-27 17:00:41
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c-Kit-IN-2 Properties

Density 1.367±0.06 g/cm3(Predicted)
storage temp. Store at -20°C
solubility Soluble in DMSO
pka 12.62±0.70(Predicted)

c-Kit-IN-2 Chemical Properties, Uses, Production

Description

c-Kit-IN-2 is a c-KIT inhibitor with an IC50 of 82 nM, shows superior antiproliferative activities against all the three GIST cell lines, GIST882, GIST430, and GIST48, with GI50s of 3, 1, and 2 nM, respectively[1]. IC50: 82 nM (c-KIT)[1]

Uses

c-Kit-IN-2 is a c-KIT inhibitor with an IC50 of 82 nM, shows superior antiproliferative activities against all the three GIST cell lines, GIST882, GIST430, and GIST48, with GI50s of 3, 1, and 2 nM, respectively[1].

References

[1]. Wu TS, et al. Discovery of Conformational Control Inhibitors Switching off the Activated c-KIT and Targeting a Broad Range of Clinically Relevant c-KIT Mutants. J Med Chem. 2019 Apr 25;62(8):3940-3957.

c-Kit-IN-2 Preparation Products And Raw materials

Raw materials

Preparation Products

c-Kit-IN-2 Suppliers

Global Suppliers ( 7)
Supplier Tel Email Country ProdList Advantage
Sichuan Wei Keqi Biological Technology Co., Ltd. 028-81700200 18116577057 3003855609@qq.com China 7717 56
BOC Sciences 16314854226; +8616314854226 inquiry@bocsci.com United States 19852 58
TargetMol Chemicals Inc. +1-781-999-5354; +1-00000000000 marketing@targetmol.com United States 32431 58
TargetMol Chemicals Inc. 15002134094 marketing@targetmol.cn China 29874 58
TargetMol Chemicals Inc. +1-781-999-5354; support@targetmol.com United States 38999 58
TargetMol Chemicals Inc. 13564774135 marketing@targetmol.com United States 19950 58
Supplier Advantage
Sichuan Wei Keqi Biological Technology Co., Ltd. 56
BOC Sciences 58
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58
TargetMol Chemicals Inc. 58

View Latest Price from c-Kit-IN-2 manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
c-Kit-IN-2 pictures 2026-07-27 c-Kit-IN-2
2121515-37-3
 $2420.00-4300.00 98.68% 10g TargetMol Chemicals Inc.
c-Kit-IN-2 pictures 2026-07-27 c-Kit-IN-2
2121515-37-3
 $2420.00-4300.00 98.68% 10g TargetMol Chemicals Inc.
c-Kit-IN-2 pictures 2025-07-23 c-Kit-IN-2
2121515-37-3
 $1670.00-2800.00 10g TargetMol Chemicals Inc.
  • c-Kit-IN-2 pictures
  • c-Kit-IN-2
    2121515-37-3
  • $2420.00-4300.00
  • 98.68%
  • TargetMol Chemicals Inc.
  • c-Kit-IN-2 pictures
  • c-Kit-IN-2
    2121515-37-3
  • $2420.00-4300.00
  • 98.68%
  • TargetMol Chemicals Inc.
  • c-Kit-IN-2 pictures
  • c-Kit-IN-2
    2121515-37-3
  • $1670.00-2800.00
  • TargetMol Chemicals Inc.

2121515-37-3 (c-Kit-IN-2) Related Search:

CD117/C-KIT Protein, HUMAN (P10721-2, HEK293, HIS) Motesanib CD117/c-kit Protein, Human (Biotinylated, HEK293, His-Avi) Sitravatinib CD117/C-KIT Protein, HUMAN (HEK293, HIS)
Dovitinib

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c-Kit-IN-2 c Kit IN 2,cKitIN2 Urea, N-(5-ethyl-3-isoxazolyl)-N'-[4-[2-[[6-(4-ethyl-1-piperazinyl)-4-pyrimidinyl]amino]-5-thiazolyl]phenyl]- 2121515-37-3