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PKG Inhibitor (trifluoroacetate salt)

CAS No.
Chemical Name:
PKG Inhibitor (trifluoroacetate salt)
Synonyms
PKG Inhibitor (trifluoroacetate salt)
CBNumber:
CB715717545
Molecular Formula:
Molecular Weight:
0
MDL Number:
MOL File:
Mol file
Last updated:2025-08-21 11:10:20

PKG Inhibitor (trifluoroacetate salt) Properties

solubility DMF: 5 mg/ml
DMSO: 15 mg/mlPBS (pH 7.2): 10 mg/ml

PKG Inhibitor (trifluoroacetate salt) price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Cayman Chemical 15995 PKG Inhibitor (trifluoroacetate salt) ≥95% 1mg $63 2026-04-30 Buy
Cayman Chemical 15995 PKG Inhibitor (trifluoroacetate salt) ≥95% 5mg $289 2026-04-30 Buy
Cayman Chemical 15995 PKG Inhibitor (trifluoroacetate salt) ≥95% 10mg $514 2026-04-30 Buy
Product number Packaging Price Buy
15995 1mg $63 Buy
15995 5mg $289 Buy
15995 10mg $514 Buy

PKG Inhibitor (trifluoroacetate salt) Chemical Properties, Uses, Production

Description

PKG inhibitor is a specific cGMP-dependent PKG inhibitor (Ki = 86 µM).1 This synthetic peptide is a nonphosphorylatable analog of a substrate corresponding to the serine-32 phosphorylation site in histone H2B.1 PKG inhibitor has been reported to block cGMP-dependent NMDA potentiation and nitric oxide-induced depression of GABA currents in cultured retinal amacrine cells.2WARNING This product is not for human or veterinary use.

References

[1] GLASS D B. Differential responses of cyclic GMP-dependent and cyclic AMP-dependent protein kinases to synthetic peptide inhibitors.[J]. Biochemical Journal, 1983, 213 1: 159-164. DOI: 10.1042/bj2130159
[2] E M WEXLER  S N  P K Stanton. Nitric oxide depresses GABAA receptor function via coactivation of cGMP-dependent kinase and phosphodiesterase.[J]. Journal of Neuroscience, 1998, 18 7: 2342-2349.

PKG Inhibitor (trifluoroacetate salt) Preparation Products And Raw materials

Raw materials

Preparation Products

PKG Inhibitor (trifluoroacetate salt) Suppliers

Global Suppliers ( 1)
Supplier Tel Email Country ProdList Advantage
Cayman Chemical Company -- sales@caymanchem.com China 6808 58
Supplier Advantage
Cayman Chemical Company 58
PKG Inhibitor (trifluoroacetate salt)