Icatibant Acetate
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- $72 - $5654.2
- Product name: Icatibant Acetate
- CAS: 138614-30-9
- MF: C59H89N19O13S.C2H4O2
- MW: 1364.59
- EINECS:206-141-6
- MDL Number:MFCD04112967
- Synonyms:HOE-140 (Icatibant);HOE140; ICATIBANT;HOE 140;CS-1399;Firazyr;HOE 140 SYNTHETIC >99% SELECTIVE B2 BRAD YKIN;d-arg-l-arg-l-pro-l-hyp-gly-l-(2-thienyl)ala-l-ser-d-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-l-(2α,3β,7aβ)-octahydro-1h-indole-2-carbonyl-l-arg;Icatibant acetate, D-Arg-L-Arg-L-Pro-L-Hyp-Gly-L-(2-thienyl)Ala-L-Ser-D-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-L-(2α,3β,7aβ)-octahydro-1H-indole-2-carbonyl-L-Arg;HOE 140 Acetate
48 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TRC
Package
- 10mM*1mLinDMSO(Solution)
- 10mM*1mLinDMSO(Solid+Solvent)
- 250μg
- 1mg
- 10mM*1mLinDMSO
- 500μg
- 2mg
- 5mg
- 10mg
- 25MG
- 50mg
- 100mg
- 250mg
- 1g
- Manufactureraablocks
- Product numberAA0018T0
- Product descriptionL-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt)
- Packaging1mg
- Price$72
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0018T0
- Product descriptionL-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt)
- Packaging2mg
- Price$99
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0018T0
- Product descriptionL-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt)
- Packaging5mg
- Price$178
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0018T0
- Product descriptionL-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) ≥98%
- Packaging50mg
- Price$189
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0018T0
- Product descriptionL-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) ≥98%
- Packaging100mg
- Price$324
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0018T0
- Product descriptionL-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) ≥98%
- Packaging250mg
- Price$551
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberZ238474
- Product descriptionIcatibant Acetate 98%
- Packaging100MG
- Price$250
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberZ238474
- Product descriptionIcatibant Acetate 98%
- Packaging25MG
- Price$125
- Updated2026-05-27
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0010072
- Product descriptionICATIBANT ACETATE 95.00%
- Packaging5MG
- Price$775
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0010072
- Product descriptionICATIBANT ACETATE 95.00%
- Packaging1MG
- Price$525
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC6403
- Product descriptionIcatibant Acetate
- Packaging1mg
- Price$90
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberC6403
- Product descriptionIcatibant Acetate
- Packaging5mg
- Price$225
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberC6403
- Product descriptionIcatibant Acetate
- Packaging25mg
- Price$620
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberC6403
- Product descriptionIcatibant Acetate
- Packaging10mg
- Price$360
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberHY-108896
- Product descriptionIcatibant acetate 99.87%
- Packaging10mg
- Price$361
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-108896
- Product descriptionIcatibant acetate 99.87%
- Packaging10mM*1mLinDMSO(Solid+Solvent)
- Price$515
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA0018T0 | L-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) | 1mg | $72 | 2026-05-28 | Buy |
| aablocks | AA0018T0 | L-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) | 2mg | $99 | 2026-05-28 | Buy |
| aablocks | AA0018T0 | L-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) | 5mg | $178 | 2026-05-28 | Buy |
| aablocks | AA0018T0 | L-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) ≥98% | 50mg | $189 | 2026-05-28 | Buy |
| aablocks | AA0018T0 | L-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) ≥98% | 100mg | $324 | 2026-05-28 | Buy |
| aablocks | AA0018T0 | L-Arginine, D-arginyl-L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-(3R)-1,2,3,4-tetrahydro-3-isoquinolinecarbonyl-(2S,3aS,7aS)-octahydro-1H-indole-2-carbonyl-, acetate (salt) ≥98% | 250mg | $551 | 2026-05-28 | Buy |
| ACHEMBLOCK | Z238474 | Icatibant Acetate 98% | 100MG | $250 | 2026-05-27 | Buy |
| ACHEMBLOCK | Z238474 | Icatibant Acetate 98% | 25MG | $125 | 2026-05-27 | Buy |
| American Custom Chemicals Corporation | API0010072 | ICATIBANT ACETATE 95.00% | 5MG | $775 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0010072 | ICATIBANT ACETATE 95.00% | 1MG | $525 | 2021-12-16 | Buy |
| ApexBio Technology | C6403 | Icatibant Acetate | 1mg | $90 | 2026-05-06 | Buy |
| ApexBio Technology | C6403 | Icatibant Acetate | 5mg | $225 | 2026-05-06 | Buy |
| ApexBio Technology | C6403 | Icatibant Acetate | 25mg | $620 | 2026-05-06 | Buy |
| ApexBio Technology | C6403 | Icatibant Acetate | 10mg | $360 | 2026-05-06 | Buy |
| Arctom | HY-108896 | Icatibant acetate 99.87% | 10mg | $361 | 2026-05-26 | Buy |
| Arctom | HY-108896 | Icatibant acetate 99.87% | 10mM*1mLinDMSO(Solid+Solvent) | $515 | 2026-05-26 | Buy |
Properties
storage temp. :-20°C
solubility :DMSO:65.0(Max Conc. mg/mL);47.63(Max Conc. mM)
Ethanol:0.25(Max Conc. mg/mL);0.18(Max Conc. mM)
PBS (pH 7.2):10.0(Max Conc. mg/mL);7.33(Max Conc. mM) form :A crystalline solid
color :White to off-white
InChIKey :HKMZRZUEADSZDQ-SUJPMXFINA-N
solubility :DMSO:65.0(Max Conc. mg/mL);47.63(Max Conc. mM)
Ethanol:0.25(Max Conc. mg/mL);0.18(Max Conc. mM)
PBS (pH 7.2):10.0(Max Conc. mg/mL);7.33(Max Conc. mM) form :A crystalline solid
color :White to off-white
InChIKey :HKMZRZUEADSZDQ-SUJPMXFINA-N
Safety Information
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Description
Although it is a rare disease, HAE is an autosomal dominant disorder that can be potentially life-threatening when swelling manifests itself within the upper airways. Antagonism of the constitutively expressed B2 receptor, therefore, would not only be beneficial in the treatment of HAE but also find application in inflammatory, allergic, and hyperalgesic disorders.Designed to possess enhanced metabolic stability with the inclusion of five non-proteinogenic amino acids, icatibant is a competitive and selective B2 receptor antagonist (devoid of activity against the inducible B1 receptor) with a Ki of 2.2±0.7 nM, and it is the first downstream targeting agent to receive regulatory approval. It joins purified C1 esterase inhibitor, danazol (an attenuated androgen), and tranexamic acid (an antifibrinolytic agent) as acute and prophylactic treatments for HAE.Related product price
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Suppliers and manufacturers
Hebei Xinsheng New Material Technology Co., LTD.
Icatibant acetate
CAS:138614-30-9
Hefei Lbao Physical & Chemical Science Co.,Ltd
Nantong Guangyuan Chemicl Co,Ltd
ATK CHEMICAL COMPANY LIMITED
BOC Sciences
Hebei Yanxi Chemical Co., Ltd.
Icatibant acetate
CAS:138614-30-9
