Telatinib
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- $55 - $2120
- Product name: Telatinib
- CAS: 332012-40-5
- MF: C20H16ClN5O3
- MW: 409.83
- EINECS:
- MDL Number:MFCD18251453
- Synonyms:2-Pyridinecarboxamide, 4-(((4-((4-chlorophenyl)amino)furo(2,3-D)pyridazin-7-yl)oxy)methyl)-N-methyl-;Bay 57-9352;Unii-18p7197Q7j;Telatinib(BAY 57-9352);4-[[[4-[(4-Chlorophenyl)amino]furo[2,3-d]pyridazin-7-yl]oxy]methyl]-N-methyl-2-pyridinecarboxamide;4-((4-(4-chlorophenylamino)furo[2,3-d]pyridazin-7-yloxy)methyl)-N-methylpicolinamide;4-[[[4-[(4-Chlorophenyl)amino]furo[2,3-d]pyridazin-7-yl]oxy]methyl]-N-methyl-2-pyridinecarboxamide Telatinib(BAY57-9352);Telatnib
32 prices
Selected condition：
Brand
- American Custom Chemicals Corporation
- ApexBio Technology
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Medical Isotopes, Inc.
- TRC
Package
- 10mM(in 1mL DMSO)
- 5MG
- 10MG
- 25mg
- 10mM(in1mLDMSO)
- 50mg
- 100MG
- 1g
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0000599
- Product descriptionTELATINIB 95.00%
- Packaging5MG
- Price$490
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0000599
- Product descriptionTELATINIB 95.00%
- Packaging10MG
- Price$739.2
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0000599
- Product descriptionTELATINIB 95.00%
- Packaging100MG
- Price$1871.1
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib(BAY57-9352)
- Packaging50mg
- Price$679
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib(BAY57-9352)
- Packaging10mg
- Price$224
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib (BAY 57-9352)
- Packaging5mg
- Price$55
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib (BAY 57-9352)
- Packaging10mM(in1mLDMSO)
- Price$66
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib (BAY 57-9352)
- Packaging10mg
- Price$77
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib(BAY57-9352)
- Packaging5mg
- Price$119
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib(BAY57-9352)
- Packaging10mM(in 1mL DMSO)
- Price$119
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8550
- Product descriptionTelatinib (BAY 57-9352)
- Packaging50mg
- Price$275
- Updated2026-05-06
- Buy
- ManufacturerCayman Chemical
- Product number26203
- Product descriptionTelatinib
- Packaging25mg
- Price$389
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number26203
- Product descriptionTelatinib ≥98%
- Packaging25mg
- Price$428
- Updated2026-04-30
- Buy
- ManufacturerCayman Chemical
- Product number26203
- Product descriptionTelatinib
- Packaging5mg
- Price$98
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number26203
- Product descriptionTelatinib ≥98%
- Packaging5mg
- Price$108
- Updated2026-04-30
- Buy
- ManufacturerCayman Chemical
- Product number26203
- Product descriptionTelatinib
- Packaging10mg
- Price$167
- Updated2024-03-01
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| American Custom Chemicals Corporation | KIN0000599 | TELATINIB 95.00% | 5MG | $490 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0000599 | TELATINIB 95.00% | 10MG | $739.2 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0000599 | TELATINIB 95.00% | 100MG | $1871.1 | 2021-12-16 | Buy |
| ApexBio Technology | A8550 | Telatinib(BAY57-9352) | 50mg | $679 | 2021-12-16 | Buy |
| ApexBio Technology | A8550 | Telatinib(BAY57-9352) | 10mg | $224 | 2021-12-16 | Buy |
| ApexBio Technology | A8550 | Telatinib (BAY 57-9352) | 5mg | $55 | 2026-05-06 | Buy |
| ApexBio Technology | A8550 | Telatinib (BAY 57-9352) | 10mM(in1mLDMSO) | $66 | 2026-05-06 | Buy |
| ApexBio Technology | A8550 | Telatinib (BAY 57-9352) | 10mg | $77 | 2026-05-06 | Buy |
| ApexBio Technology | A8550 | Telatinib(BAY57-9352) | 5mg | $119 | 2021-12-16 | Buy |
| ApexBio Technology | A8550 | Telatinib(BAY57-9352) | 10mM(in 1mL DMSO) | $119 | 2021-12-16 | Buy |
| ApexBio Technology | A8550 | Telatinib (BAY 57-9352) | 50mg | $275 | 2026-05-06 | Buy |
| Cayman Chemical | 26203 | Telatinib | 25mg | $389 | 2024-03-01 | Buy |
| Cayman Chemical | 26203 | Telatinib ≥98% | 25mg | $428 | 2026-04-30 | Buy |
| Cayman Chemical | 26203 | Telatinib | 5mg | $98 | 2024-03-01 | Buy |
| Cayman Chemical | 26203 | Telatinib ≥98% | 5mg | $108 | 2026-04-30 | Buy |
| Cayman Chemical | 26203 | Telatinib | 10mg | $167 | 2024-03-01 | Buy |
Properties
Boiling point :713.6±60.0 °C(Predicted)
Density :1.417
storage temp. :Store at -20°C
solubility :insoluble in H2O; insoluble in EtOH; ≥20.5 mg/mL in DMSO
form :solid
pka :14.18±0.46(Predicted)
color :White to light yellow
InChI :InChI=1S/C20H16ClN5O3/c1-22-19(27)16-10-12(6-8-23-16)11-29-20-17-15(7-9-28-17)18(25-26-20)24-14-4-2-13(21)3-5-14/h2-10H,11H2,1H3,(H,22,27)(H,24,25)
InChIKey :QFCXANHHBCGMAS-UHFFFAOYSA-N
SMILES :C1(C(NC)=O)=NC=CC(COC2=NN=C(NC3=CC=C(Cl)C=C3)C3C=COC2=3)=C1
Density :1.417
storage temp. :Store at -20°C
solubility :insoluble in H2O; insoluble in EtOH; ≥20.5 mg/mL in DMSO
form :solid
pka :14.18±0.46(Predicted)
color :White to light yellow
InChI :InChI=1S/C20H16ClN5O3/c1-22-19(27)16-10-12(6-8-23-16)11-29-20-17-15(7-9-28-17)18(25-26-20)24-14-4-2-13(21)3-5-14/h2-10H,11H2,1H3,(H,22,27)(H,24,25)
InChIKey :QFCXANHHBCGMAS-UHFFFAOYSA-N
SMILES :C1(C(NC)=O)=NC=CC(COC2=NN=C(NC3=CC=C(Cl)C=C3)C3C=COC2=3)=C1
Safety Information
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Description
Telatinib is a multi-kinase inhibitor that inhibits VEGF receptor 2 (VEGFR2), VEGFR3, PDGFRα, and c-Kit (IC50s = 6, 4, 15, and 1 nM, respectively). It also binds to the transmembrane region of the ABCG2 efflux transporter and enhances intracellular accumulation of [3H]-mitoxantrone in ABCG2-overexpressing cells. Telatinib (15 mg/kg) decreases tumor growth rate and size in an H460/MX20 mouse xenograft model.More related product prices
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