pristimerin
|
- $47 - $2690
- Product name: pristimerin
- CAS: 1258-84-0
- MF: C30H40O4
- MW: 464.64
- EINECS:251-228-4
- MDL Number:MFCD01711331
- Synonyms:pristimerin;3-Hydroxy-2-oxo-24-nor-D:A-friedoolean-1(10),3,5,7-tetren-29-oic acid methyl ester;Celastrol-methylether;(9β,13α,14β,20α)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oicacidmethylester;(9b,13a,14b,20a)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tertraen-29-oic acid methyl ester;3-hydroxy-9β,13α-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid, methyl ester;Celastrol methyl ester;Pristimerin(NSC 99281)
58 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- JR MediChem
- Medical Isotopes, Inc.
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 10
- 1mg
- 5mg
- 1mlx10mM(inDMSO)
- 10mg
- 20mg
- 25mg
- 50mg
- 100mg
- 250mg
- 500mg
- 1000mg
- 1g
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin
- Packaging1mg
- Price$47
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin ≥98%(HPLC)
- Packaging5mg
- Price$67
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin ≥98%(HPLC)
- Packaging10mg
- Price$120
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin
- Packaging25mg
- Price$255
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin 95%
- Packaging50mg
- Price$342
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin 95%
- Packaging100mg
- Price$558
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin 95%
- Packaging250mg
- Price$1098
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA003TVT
- Product descriptionPristimerin 95%
- Packaging1g
- Price$2690
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberU106589
- Product descriptionPristimerin 98.00%
- Packaging100MG
- Price$195
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberU106589
- Product descriptionPristimerin 98.00%
- Packaging50MG
- Price$115
- Updated2026-05-27
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006380
- Product descriptionPristimerin 95.00%
- Packaging5MG
- Price$212.3
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006380
- Product descriptionPristimerin 95.00%
- Packaging50MG
- Price$1515.94
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006380
- Product descriptionPristimerin 95.00%
- Packaging10MG
- Price$776.16
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB7488
- Product descriptionPristimerin
- Packaging50mg
- Price$530
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB7488
- Product descriptionPristimerin
- Packaging10mg
- Price$130
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberAB1292
- Product descriptionPristimerin 98%(HPLC)
- Packaging20mg
- Price$132
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA003TVT | Pristimerin | 1mg | $47 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin ≥98%(HPLC) | 5mg | $67 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin ≥98%(HPLC) | 10mg | $120 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin | 25mg | $255 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin 95% | 50mg | $342 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin 95% | 100mg | $558 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin 95% | 250mg | $1098 | 2026-05-28 | Buy |
| aablocks | AA003TVT | Pristimerin 95% | 1g | $2690 | 2026-05-28 | Buy |
| ACHEMBLOCK | U106589 | Pristimerin 98.00% | 100MG | $195 | 2026-05-27 | Buy |
| ACHEMBLOCK | U106589 | Pristimerin 98.00% | 50MG | $115 | 2026-05-27 | Buy |
| American Custom Chemicals Corporation | API0006380 | Pristimerin 95.00% | 5MG | $212.3 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006380 | Pristimerin 95.00% | 50MG | $1515.94 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006380 | Pristimerin 95.00% | 10MG | $776.16 | 2021-12-16 | Buy |
| ApexBio Technology | B7488 | Pristimerin | 50mg | $530 | 2026-05-06 | Buy |
| ApexBio Technology | B7488 | Pristimerin | 10mg | $130 | 2026-05-06 | Buy |
| Arctom | AB1292 | Pristimerin 98%(HPLC) | 20mg | $132 | 2026-05-26 | Buy |
Properties
Melting point :219.5°C
Boiling point :488.1°C (rough estimate)
Density :1.0271 (rough estimate)
refractive index :1.4800 (estimate)
storage temp. :-20°C
solubility :DMSO: ≥5mg/mL
form :Red solid
pka :8.60±0.70(Predicted)
color :orange
InChIKey :JFACETXYABVHFD-VXTIGNJVNA-N
SMILES :[C@]12(C)CC[C@@]3(C)CC[C@@](C)(C(=O)OC)C[C@@]3([H])[C@]1(C)CC[C@@]1(C)C3=CC(C(O)=C(C)C3=CC=C21)=O |&1:0,4,8,15,17,21,r|
Boiling point :488.1°C (rough estimate)
Density :1.0271 (rough estimate)
refractive index :1.4800 (estimate)
storage temp. :-20°C
solubility :DMSO: ≥5mg/mL
form :Red solid
pka :8.60±0.70(Predicted)
color :orange
InChIKey :JFACETXYABVHFD-VXTIGNJVNA-N
SMILES :[C@]12(C)CC[C@@]3(C)CC[C@@](C)(C(=O)OC)C[C@@]3([H])[C@]1(C)CC[C@@]1(C)C3=CC(C(O)=C(C)C3=CC=C21)=O |&1:0,4,8,15,17,21,r|
Safety Information
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Description
Monoacylglycerol lipase (MAGL) hydrolyzes the endogenous cannabinoid 2-arachidonoyl glycerol (2-AG), terminating its capacity to activate cannabinoid receptors. Pristimerin is a naturally occurring terpenoid that potently inhibits MAGL (IC50 = 93 nM). Its actions are rapid, reversible, and noncompetitive. Pristimerin (1 μM) significantly increases 2-AG levels in isolated rat neurons, indicating that it inhibits endogenous MAGL in cultured cells. Moreover, it does not increase levels of palmitoyl ethanolamide, suggesting that pristimerin does not affect the activity of fatty acid amide hydrolase (FAAH).More related product prices
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Suppliers and manufacturers
Huzhou ZhanShu Biotechnology Co.,Ltd
Nanjing Spring & Autumn Biological Engineering Co., Ltd.
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Chembest Research Laboratories Limited
ShangHai YuanYe Biotechnology Co., Ltd.
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Chengdu Climax Biotech Co., Ltd.
Shanghai Winherb Medical Technology Co., Ltd.
Shanghai Tauto Biotech Co., Ltd.