阻害剤活性化剤

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Structure Chemical Name CAS MF
VILAZODONE (SSRI inhibitor) VILAZODONE (SSRI inhibitor)
GSK126 (EZH2 inhibitor) GSK126 (EZH2 inhibitor)
DEGRASYN (BCR-ABL inhibitor) DEGRASYN (BCR-ABL inhibitor)
IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor) IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
DAPT (Γ-SECRETASE inhibitor) DAPT (Γ-SECRETASE inhibitor)
BLU-9931 (FGFR inhibitor) BLU-9931 (FGFR inhibitor)
ABT-199 (BCL-2 inhibitor) ABT-199 (BCL-2 inhibitor)
BYL719 (PI3K inhibitor) BYL719 (PI3K inhibitor)
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor) VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
DEFACTINIB (FAK inhibitor) DEFACTINIB (FAK inhibitor)
KU0063794 (MTOR inhibitor) KU0063794 (MTOR inhibitor)
EVEROLIMUS (MTOR inhibitor) EVEROLIMUS (MTOR inhibitor)
SALUBRINAL (PERK inhibitor) SALUBRINAL (PERK inhibitor)
FIPI (PLD1/2 inhibitor) FIPI (PLD1/2 inhibitor)
PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist) PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist)
PLX4032 (RAF inhibitor) PLX4032 (RAF inhibitor)
RNasin Inhibitor (Ribonuclease Inhibitor)) RNasin Inhibitor (Ribonuclease Inhibitor))
PD123319 (RAAS inhibitor) PD123319 (RAAS inhibitor)
A83-01 (ALK5 inhibitor) A83-01 (ALK5 inhibitor)
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor) VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
PRT062607 HCL (SYK inhibitor) PRT062607 HCL (SYK inhibitor)
BATIMASTAT (MMP inhibitor) BATIMASTAT (MMP inhibitor)
VOLASERTIB (PLK inhibitor) VOLASERTIB (PLK inhibitor)
SC-514 (IΚB/IKK inhibitor) SC-514 (IΚB/IKK inhibitor)
HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride Cl2H8N2O2
ZOTAROLIMUS (MTOR inhibitor) ZOTAROLIMUS (MTOR inhibitor)
EPZ-6438 (E7438) (EZH2 inhibitor) EPZ-6438 (E7438) (EZH2 inhibitor)
PFI-4 (EPIGENETIC READER DOMAIN inhibitor) PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
INDIPLON (GABA RECEPTOR Conditioner) INDIPLON (GABA RECEPTOR Conditioner)
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor) SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
TIVOZANIB (VEGFR inhibitor) TIVOZANIB (VEGFR inhibitor)
LINIFANIB (VEGFR inhibitor) LINIFANIB (VEGFR inhibitor)
ENTOSPLETINIB (SYK inhibitor) ENTOSPLETINIB (SYK inhibitor)
BI2536 (PLK inhibitor) BI2536 (PLK inhibitor)
AG14361 (PARP1 inhibitor) AG14361 (PARP1 inhibitor)
EG-011 EG-011 2377113-41-0 C28H26N4O4
ROMIDEPSIN (HDAC inhibitor) ROMIDEPSIN (HDAC inhibitor)
DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor) DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
PONATINIB (SRC-ABL inhibitor) PONATINIB (SRC-ABL inhibitor)
ML323 (DUB inhibitor) ML323 (DUB inhibitor)
ML141 (RHO inhibitor) ML141 (RHO inhibitor)
DACLATASVIR (HCV NS5A inhibitor) DACLATASVIR (HCV NS5A inhibitor)
PAC-1 (CASPASE Activator) PAC-1 (CASPASE Activator)
CYT997 (LEXIBULIN) (MICROTUBULES inhibitor) CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
RIMONABANT (CANNABINOID RECEPTOR antagonist) RIMONABANT (CANNABINOID RECEPTOR antagonist)
AG1024 (IGF-1R inhibitor) AG1024 (IGF-1R inhibitor)
ABT-737 (BCL-2 inhibitor) ABT-737 (BCL-2 inhibitor)
SRT 2104 (SIRT1 activator) SRT 2104 (SIRT1 activator)
TG101348 (JAK inhibitor) TG101348 (JAK inhibitor)
ICA 069673 ICA 069673 582323-16-8 C11H6ClF2N3O
(-)-BLEBBISTATIN (ATPASE inhibitor) (-)-BLEBBISTATIN (ATPASE inhibitor)
ポルフィロマイシン ポルフィロマイシン 801-52-5 C16H20N4O5
PI-103 (PI3K inhibitor) PI-103 (PI3K inhibitor)
I-BET-762 (GSK525762) (BET inhibitor) I-BET-762 (GSK525762) (BET inhibitor)
BTdCPU BTdCPU 1257423-87-2 C13H8Cl2N4OS
NECROSTATIN-1 (TNF-ALPHA inhibitor) NECROSTATIN-1 (TNF-ALPHA inhibitor)
PLERIXAFOR (CXCR inhibitor) PLERIXAFOR (CXCR inhibitor)
RG108 (DNA METHYLTRANSFERASE inhibitor) RG108 (DNA METHYLTRANSFERASE inhibitor)
B-AP15 (DUB inhibitor) B-AP15 (DUB inhibitor)
REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor) REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
IONOMYCIN (calcium ionophore) IONOMYCIN (calcium ionophore)
ODANACATIB (CYSTEINE PROTEASE inhibitor) ODANACATIB (CYSTEINE PROTEASE inhibitor)
BARDOXOLONE METHYL (IΚB/IKK inhibitor) BARDOXOLONE METHYL (IΚB/IKK inhibitor)
ISRIB (PERK inhibitor) ISRIB (PERK inhibitor)
DBEQ (P97 inhibitor) DBEQ (P97 inhibitor)
タフトシン タフトシン 9063-57-4 C21H40N8O6
KN-93 PHOSPHATE (CAMK Inhibitor) KN-93 PHOSPHATE (CAMK Inhibitor)
SALIRASIB (RHO inhibitor) SALIRASIB (RHO inhibitor)
EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor) EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
MI-2 (HISTONE METHYLTRANSFERASE Inhibitor) MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
SEMAGACESTAT (GAMMA - SECRETASE Inhibitor) SEMAGACESTAT (GAMMA - SECRETASE Inhibitor)
BMS-5 (LIMK inhibitor) BMS-5 (LIMK inhibitor)
DACOMITINIB (EGFR inhibitor) DACOMITINIB (EGFR inhibitor)
AVASIMIBE (P450 inhibitor) AVASIMIBE (P450 inhibitor)
SRT 1720 (SIRT1 activator) SRT 1720 (SIRT1 activator)
PND-1186 (FAK inhibitor) PND-1186 (FAK inhibitor)
ENZALUTAMIDE (MDV3100) (AR inhibitor) ENZALUTAMIDE (MDV3100) (AR inhibitor)
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor) COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist) BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist)
AR-A014418 (GSK-3 inhibitor) AR-A014418 (GSK-3 inhibitor)
DALCETRAPIB (CETP inhibitor) DALCETRAPIB (CETP inhibitor)
DABRAFENIB (RAF inhibitor) DABRAFENIB (RAF inhibitor)
GSK1278863 (HIF inhibitor) GSK1278863 (HIF inhibitor)
JNJ-7777120 (HISTAMINE RECEPTOR antagonist) JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
KU-55933 (ATM inhibitor) KU-55933 (ATM inhibitor)
TWS119 (GSK-3 inhibitor) TWS119 (GSK-3 inhibitor)
[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate [oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate 193743-89-4
PFI-3 (EPIGENETIC READER DOMAIN inhibitor) PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
BAY87-2243 (HIF inhibitor) BAY87-2243 (HIF inhibitor)
TEDIZOLID (MAO-A inhibitor) TEDIZOLID (MAO-A inhibitor)
TPA Deficient Plasma TPA Deficient Plasma
FK-506 (MTOR inhibitor) FK-506 (MTOR inhibitor)
TBA-354 (anti-tuberculosis) TBA-354 (anti-tuberculosis)
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor) PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
GELDANAMYCIN (HSP90 inhibitor) GELDANAMYCIN (HSP90 inhibitor)
SP600125 (JNK inhibitor) SP600125 (JNK inhibitor)
FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor) FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
INH1 (MICROTUBULE ASSOCIATED inhibitor) INH1 (MICROTUBULE ASSOCIATED inhibitor)
BML-210 (HDAC inhibitor) BML-210 (HDAC inhibitor)
OSU-03012 (PDK-1 inhibitor) OSU-03012 (PDK-1 inhibitor)
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