阻害剤活性化剤

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Structure Chemical Name CAS MF
SALUBRINAL (PERK inhibitor) SALUBRINAL (PERK inhibitor)
BLU-9931 (FGFR inhibitor) BLU-9931 (FGFR inhibitor)
ODANACATIB (CYSTEINE PROTEASE inhibitor) ODANACATIB (CYSTEINE PROTEASE inhibitor)
TBA-354 (anti-tuberculosis) TBA-354 (anti-tuberculosis)
PRT062607 HCL (SYK inhibitor) PRT062607 HCL (SYK inhibitor)
JNJ-7777120 (HISTAMINE RECEPTOR antagonist) JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
GSK126 (EZH2 inhibitor) GSK126 (EZH2 inhibitor)
SALIRASIB (RHO inhibitor) SALIRASIB (RHO inhibitor)
EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor) EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
KU0063794 (MTOR inhibitor) KU0063794 (MTOR inhibitor)
DEFACTINIB (FAK inhibitor) DEFACTINIB (FAK inhibitor)
ENTOSPLETINIB (SYK inhibitor) ENTOSPLETINIB (SYK inhibitor)
IONOMYCIN (calcium ionophore) IONOMYCIN (calcium ionophore)
(-)-BLEBBISTATIN (ATPASE inhibitor) (-)-BLEBBISTATIN (ATPASE inhibitor)
BYL719 (PI3K inhibitor) BYL719 (PI3K inhibitor)
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor) VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
LINIFANIB (VEGFR inhibitor) LINIFANIB (VEGFR inhibitor)
ROMIDEPSIN (HDAC inhibitor) ROMIDEPSIN (HDAC inhibitor)
DALCETRAPIB (CETP inhibitor) DALCETRAPIB (CETP inhibitor)
PND-1186 (FAK inhibitor) PND-1186 (FAK inhibitor)
ZOTAROLIMUS (MTOR inhibitor) ZOTAROLIMUS (MTOR inhibitor)
TG101348 (JAK inhibitor) TG101348 (JAK inhibitor)
PLX4032 (RAF inhibitor) PLX4032 (RAF inhibitor)
DAPT (Γ-SECRETASE inhibitor) DAPT (Γ-SECRETASE inhibitor)
ENZALUTAMIDE (MDV3100) (AR inhibitor) ENZALUTAMIDE (MDV3100) (AR inhibitor)
REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor) REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
BI2536 (PLK inhibitor) BI2536 (PLK inhibitor)
DEGRASYN (BCR-ABL inhibitor) DEGRASYN (BCR-ABL inhibitor)
B-AP15 (DUB inhibitor) B-AP15 (DUB inhibitor)
AVASIMIBE (P450 inhibitor) AVASIMIBE (P450 inhibitor)
PFI-4 (EPIGENETIC READER DOMAIN inhibitor) PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
FK-506 (MTOR inhibitor) FK-506 (MTOR inhibitor)
A83-01 (ALK5 inhibitor) A83-01 (ALK5 inhibitor)
VILAZODONE (SSRI inhibitor) VILAZODONE (SSRI inhibitor)
KU-55933 (ATM inhibitor) KU-55933 (ATM inhibitor)
VOLASERTIB (PLK inhibitor) VOLASERTIB (PLK inhibitor)
EVEROLIMUS (MTOR inhibitor) EVEROLIMUS (MTOR inhibitor)
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor) VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate [oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate 193743-89-4
PI-103 (PI3K inhibitor) PI-103 (PI3K inhibitor)
I-BET-762 (GSK525762) (BET inhibitor) I-BET-762 (GSK525762) (BET inhibitor)
ABT-199 (BCL-2 inhibitor) ABT-199 (BCL-2 inhibitor)
ポルフィロマイシン ポルフィロマイシン 801-52-5 C16H20N4O5
PONATINIB (SRC-ABL inhibitor) PONATINIB (SRC-ABL inhibitor)
ML323 (DUB inhibitor) ML323 (DUB inhibitor)
DABRAFENIB (RAF inhibitor) DABRAFENIB (RAF inhibitor)
GSK1278863 (HIF inhibitor) GSK1278863 (HIF inhibitor)
ISRIB (PERK inhibitor) ISRIB (PERK inhibitor)
IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor) IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
タフトシン タフトシン 9063-57-4 C21H40N8O6
SRT 1720 (SIRT1 activator) SRT 1720 (SIRT1 activator)
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor) COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist) BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist)
RG108 (DNA METHYLTRANSFERASE inhibitor) RG108 (DNA METHYLTRANSFERASE inhibitor)
EG-011 EG-011 2377113-41-0 C28H26N4O4
TIVOZANIB (VEGFR inhibitor) TIVOZANIB (VEGFR inhibitor)
KN-93 PHOSPHATE (CAMK Inhibitor) KN-93 PHOSPHATE (CAMK Inhibitor)
GELDANAMYCIN (HSP90 inhibitor) GELDANAMYCIN (HSP90 inhibitor)
SP600125 (JNK inhibitor) SP600125 (JNK inhibitor)
PFI-3 (EPIGENETIC READER DOMAIN inhibitor) PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
BAY87-2243 (HIF inhibitor) BAY87-2243 (HIF inhibitor)
PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist) PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist)
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor) SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
BML-210 (HDAC inhibitor) BML-210 (HDAC inhibitor)
OSU-03012 (PDK-1 inhibitor) OSU-03012 (PDK-1 inhibitor)
AG14361 (PARP1 inhibitor) AG14361 (PARP1 inhibitor)
DBEQ (P97 inhibitor) DBEQ (P97 inhibitor)
MI-2 (HISTONE METHYLTRANSFERASE Inhibitor) MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
SEMAGACESTAT (GAMMA - SECRETASE Inhibitor) SEMAGACESTAT (GAMMA - SECRETASE Inhibitor)
INDIPLON (GABA RECEPTOR Conditioner) INDIPLON (GABA RECEPTOR Conditioner)
ICA 069673 ICA 069673 582323-16-8 C11H6ClF2N3O
AR-A014418 (GSK-3 inhibitor) AR-A014418 (GSK-3 inhibitor)
DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor) DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
PAC-1 (CASPASE Activator) PAC-1 (CASPASE Activator)
TPA Deficient Plasma TPA Deficient Plasma
RNasin Inhibitor (Ribonuclease Inhibitor)) RNasin Inhibitor (Ribonuclease Inhibitor))
PD123319 (RAAS inhibitor) PD123319 (RAAS inhibitor)
BARDOXOLONE METHYL (IΚB/IKK inhibitor) BARDOXOLONE METHYL (IΚB/IKK inhibitor)
RIMONABANT (CANNABINOID RECEPTOR antagonist) RIMONABANT (CANNABINOID RECEPTOR antagonist)
AG1024 (IGF-1R inhibitor) AG1024 (IGF-1R inhibitor)
BMS-5 (LIMK inhibitor) BMS-5 (LIMK inhibitor)
DACOMITINIB (EGFR inhibitor) DACOMITINIB (EGFR inhibitor)
BTdCPU BTdCPU 1257423-87-2 C13H8Cl2N4OS
TEDIZOLID (MAO-A inhibitor) TEDIZOLID (MAO-A inhibitor)
PLERIXAFOR (CXCR inhibitor) PLERIXAFOR (CXCR inhibitor)
HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride Cl2H8N2O2
FIPI (PLD1/2 inhibitor) FIPI (PLD1/2 inhibitor)
ABT-737 (BCL-2 inhibitor) ABT-737 (BCL-2 inhibitor)
CYT997 (LEXIBULIN) (MICROTUBULES inhibitor) CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
TWS119 (GSK-3 inhibitor) TWS119 (GSK-3 inhibitor)
U-104 (CARBONIC ANHYDRASE INHIBITOR) U-104 (CARBONIC ANHYDRASE INHIBITOR)
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor) PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
EPZ-6438 (E7438) (EZH2 inhibitor) EPZ-6438 (E7438) (EZH2 inhibitor)
SC-514 (IΚB/IKK inhibitor) SC-514 (IΚB/IKK inhibitor)
FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor) FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
SRT 2104 (SIRT1 activator) SRT 2104 (SIRT1 activator)
NECROSTATIN-1 (TNF-ALPHA inhibitor) NECROSTATIN-1 (TNF-ALPHA inhibitor)
INH1 (MICROTUBULE ASSOCIATED inhibitor) INH1 (MICROTUBULE ASSOCIATED inhibitor)
ML141 (RHO inhibitor) ML141 (RHO inhibitor)
DACLATASVIR (HCV NS5A inhibitor) DACLATASVIR (HCV NS5A inhibitor)
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