阻害剤活性化剤

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Structure Chemical Name CAS MF
RG108 (DNA METHYLTRANSFERASE inhibitor) RG108 (DNA METHYLTRANSFERASE inhibitor)
DACOMITINIB (EGFR inhibitor) DACOMITINIB (EGFR inhibitor)
ODANACATIB (CYSTEINE PROTEASE inhibitor) ODANACATIB (CYSTEINE PROTEASE inhibitor)
TBA-354 (anti-tuberculosis) TBA-354 (anti-tuberculosis)
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor) PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
ENTOSPLETINIB (SYK inhibitor) ENTOSPLETINIB (SYK inhibitor)
DACLATASVIR (HCV NS5A inhibitor) DACLATASVIR (HCV NS5A inhibitor)
TWS119 (GSK-3 inhibitor) TWS119 (GSK-3 inhibitor)
U-104 (CARBONIC ANHYDRASE INHIBITOR) U-104 (CARBONIC ANHYDRASE INHIBITOR)
PRT062607 HCL (SYK inhibitor) PRT062607 HCL (SYK inhibitor)
HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride Cl2H8N2O2
FIPI (PLD1/2 inhibitor) FIPI (PLD1/2 inhibitor)
PI-103 (PI3K inhibitor) PI-103 (PI3K inhibitor)
BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist) BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist)
NECROSTATIN-1 (TNF-ALPHA inhibitor) NECROSTATIN-1 (TNF-ALPHA inhibitor)
SRT 2104 (SIRT1 activator) SRT 2104 (SIRT1 activator)
RNasin Inhibitor (Ribonuclease Inhibitor)) RNasin Inhibitor (Ribonuclease Inhibitor))
PD123319 (RAAS inhibitor) PD123319 (RAAS inhibitor)
BARDOXOLONE METHYL (IΚB/IKK inhibitor) BARDOXOLONE METHYL (IΚB/IKK inhibitor)
DEGRASYN (BCR-ABL inhibitor) DEGRASYN (BCR-ABL inhibitor)
IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor) IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
DABRAFENIB (RAF inhibitor) DABRAFENIB (RAF inhibitor)
EG-011 EG-011 2377113-41-0 C28H26N4O4
VILAZODONE (SSRI inhibitor) VILAZODONE (SSRI inhibitor)
KU-55933 (ATM inhibitor) KU-55933 (ATM inhibitor)
AR-A014418 (GSK-3 inhibitor) AR-A014418 (GSK-3 inhibitor)
DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor) DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
ROMIDEPSIN (HDAC inhibitor) ROMIDEPSIN (HDAC inhibitor)
DALCETRAPIB (CETP inhibitor) DALCETRAPIB (CETP inhibitor)
TG101348 (JAK inhibitor) TG101348 (JAK inhibitor)
PLX4032 (RAF inhibitor) PLX4032 (RAF inhibitor)
JNJ-7777120 (HISTAMINE RECEPTOR antagonist) JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
GSK126 (EZH2 inhibitor) GSK126 (EZH2 inhibitor)
BMS-5 (LIMK inhibitor) BMS-5 (LIMK inhibitor)
GSK1278863 (HIF inhibitor) GSK1278863 (HIF inhibitor)
PONATINIB (SRC-ABL inhibitor) PONATINIB (SRC-ABL inhibitor)
ML323 (DUB inhibitor) ML323 (DUB inhibitor)
ISRIB (PERK inhibitor) ISRIB (PERK inhibitor)
B-AP15 (DUB inhibitor) B-AP15 (DUB inhibitor)
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor) VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate [oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate 193743-89-4
VOLASERTIB (PLK inhibitor) VOLASERTIB (PLK inhibitor)
EVEROLIMUS (MTOR inhibitor) EVEROLIMUS (MTOR inhibitor)
REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor) REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
IONOMYCIN (calcium ionophore) IONOMYCIN (calcium ionophore)
FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor) FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
INH1 (MICROTUBULE ASSOCIATED inhibitor) INH1 (MICROTUBULE ASSOCIATED inhibitor)
INDIPLON (GABA RECEPTOR Conditioner) INDIPLON (GABA RECEPTOR Conditioner)
SEMAGACESTAT (GAMMA - SECRETASE Inhibitor) SEMAGACESTAT (GAMMA - SECRETASE Inhibitor)
DAPT (Γ-SECRETASE inhibitor) DAPT (Γ-SECRETASE inhibitor)
ENZALUTAMIDE (MDV3100) (AR inhibitor) ENZALUTAMIDE (MDV3100) (AR inhibitor)
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor) VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
LINIFANIB (VEGFR inhibitor) LINIFANIB (VEGFR inhibitor)
(-)-BLEBBISTATIN (ATPASE inhibitor) (-)-BLEBBISTATIN (ATPASE inhibitor)
BYL719 (PI3K inhibitor) BYL719 (PI3K inhibitor)
SALIRASIB (RHO inhibitor) SALIRASIB (RHO inhibitor)
BI2536 (PLK inhibitor) BI2536 (PLK inhibitor)
BTdCPU BTdCPU 1257423-87-2 C13H8Cl2N4OS
TEDIZOLID (MAO-A inhibitor) TEDIZOLID (MAO-A inhibitor)
PLERIXAFOR (CXCR inhibitor) PLERIXAFOR (CXCR inhibitor)
AG14361 (PARP1 inhibitor) AG14361 (PARP1 inhibitor)
DBEQ (P97 inhibitor) DBEQ (P97 inhibitor)
タフトシン タフトシン 9063-57-4 C21H40N8O6
SRT 1720 (SIRT1 activator) SRT 1720 (SIRT1 activator)
RIMONABANT (CANNABINOID RECEPTOR antagonist) RIMONABANT (CANNABINOID RECEPTOR antagonist)
AG1024 (IGF-1R inhibitor) AG1024 (IGF-1R inhibitor)
TIVOZANIB (VEGFR inhibitor) TIVOZANIB (VEGFR inhibitor)
KN-93 PHOSPHATE (CAMK Inhibitor) KN-93 PHOSPHATE (CAMK Inhibitor)
BML-210 (HDAC inhibitor) BML-210 (HDAC inhibitor)
CYT997 (LEXIBULIN) (MICROTUBULES inhibitor) CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist) PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist)
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor) SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
FK-506 (MTOR inhibitor) FK-506 (MTOR inhibitor)
A83-01 (ALK5 inhibitor) A83-01 (ALK5 inhibitor)
SALUBRINAL (PERK inhibitor) SALUBRINAL (PERK inhibitor)
BLU-9931 (FGFR inhibitor) BLU-9931 (FGFR inhibitor)
AVASIMIBE (P450 inhibitor) AVASIMIBE (P450 inhibitor)
I-BET-762 (GSK525762) (BET inhibitor) I-BET-762 (GSK525762) (BET inhibitor)
PAC-1 (CASPASE Activator) PAC-1 (CASPASE Activator)
TPA Deficient Plasma TPA Deficient Plasma
PND-1186 (FAK inhibitor) PND-1186 (FAK inhibitor)
ZOTAROLIMUS (MTOR inhibitor) ZOTAROLIMUS (MTOR inhibitor)
PFI-3 (EPIGENETIC READER DOMAIN inhibitor) PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
BAY87-2243 (HIF inhibitor) BAY87-2243 (HIF inhibitor)
ABT-199 (BCL-2 inhibitor) ABT-199 (BCL-2 inhibitor)
EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor) EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
ML141 (RHO inhibitor) ML141 (RHO inhibitor)
ポルフィロマイシン ポルフィロマイシン 801-52-5 C16H20N4O5
EPZ-6438 (E7438) (EZH2 inhibitor) EPZ-6438 (E7438) (EZH2 inhibitor)
SC-514 (IΚB/IKK inhibitor) SC-514 (IΚB/IKK inhibitor)
MI-2 (HISTONE METHYLTRANSFERASE Inhibitor) MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
ICA 069673 ICA 069673 582323-16-8 C11H6ClF2N3O
KU0063794 (MTOR inhibitor) KU0063794 (MTOR inhibitor)
DEFACTINIB (FAK inhibitor) DEFACTINIB (FAK inhibitor)
ABT-737 (BCL-2 inhibitor) ABT-737 (BCL-2 inhibitor)
OSU-03012 (PDK-1 inhibitor) OSU-03012 (PDK-1 inhibitor)
GELDANAMYCIN (HSP90 inhibitor) GELDANAMYCIN (HSP90 inhibitor)
SP600125 (JNK inhibitor) SP600125 (JNK inhibitor)
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor) COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
PFI-4 (EPIGENETIC READER DOMAIN inhibitor) PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
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