阻害剤活性化剤

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Structure Chemical Name CAS MF
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor) VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
U-104 (CARBONIC ANHYDRASE INHIBITOR) U-104 (CARBONIC ANHYDRASE INHIBITOR)
PRT062607 HCL (SYK inhibitor) PRT062607 HCL (SYK inhibitor)
VOLASERTIB (PLK inhibitor) VOLASERTIB (PLK inhibitor)
EVEROLIMUS (MTOR inhibitor) EVEROLIMUS (MTOR inhibitor)
DABRAFENIB (RAF inhibitor) DABRAFENIB (RAF inhibitor)
EG-011 EG-011 2377113-41-0 C28H26N4O4
RNasin Inhibitor (Ribonuclease Inhibitor)) RNasin Inhibitor (Ribonuclease Inhibitor))
PD123319 (RAAS inhibitor) PD123319 (RAAS inhibitor)
BARDOXOLONE METHYL (IΚB/IKK inhibitor) BARDOXOLONE METHYL (IΚB/IKK inhibitor)
TWS119 (GSK-3 inhibitor) TWS119 (GSK-3 inhibitor)
TBA-354 (anti-tuberculosis) TBA-354 (anti-tuberculosis)
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor) PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
(-)-BLEBBISTATIN (ATPASE inhibitor) (-)-BLEBBISTATIN (ATPASE inhibitor)
DACLATASVIR (HCV NS5A inhibitor) DACLATASVIR (HCV NS5A inhibitor)
KU0063794 (MTOR inhibitor) KU0063794 (MTOR inhibitor)
DEFACTINIB (FAK inhibitor) DEFACTINIB (FAK inhibitor)
ISRIB (PERK inhibitor) ISRIB (PERK inhibitor)
B-AP15 (DUB inhibitor) B-AP15 (DUB inhibitor)
DAPT (Γ-SECRETASE inhibitor) DAPT (Γ-SECRETASE inhibitor)
KU-55933 (ATM inhibitor) KU-55933 (ATM inhibitor)
SALIRASIB (RHO inhibitor) SALIRASIB (RHO inhibitor)
BI2536 (PLK inhibitor) BI2536 (PLK inhibitor)
RG108 (DNA METHYLTRANSFERASE inhibitor) RG108 (DNA METHYLTRANSFERASE inhibitor)
GSK1278863 (HIF inhibitor) GSK1278863 (HIF inhibitor)
PND-1186 (FAK inhibitor) PND-1186 (FAK inhibitor)
ZOTAROLIMUS (MTOR inhibitor) ZOTAROLIMUS (MTOR inhibitor)
ABT-737 (BCL-2 inhibitor) ABT-737 (BCL-2 inhibitor)
OSU-03012 (PDK-1 inhibitor) OSU-03012 (PDK-1 inhibitor)
JNJ-7777120 (HISTAMINE RECEPTOR antagonist) JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
GSK126 (EZH2 inhibitor) GSK126 (EZH2 inhibitor)
AVASIMIBE (P450 inhibitor) AVASIMIBE (P450 inhibitor)
KN-93 PHOSPHATE (CAMK Inhibitor) KN-93 PHOSPHATE (CAMK Inhibitor)
BML-210 (HDAC inhibitor) BML-210 (HDAC inhibitor)
CYT997 (LEXIBULIN) (MICROTUBULES inhibitor) CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
VILAZODONE (SSRI inhibitor) VILAZODONE (SSRI inhibitor)
BLU-9931 (FGFR inhibitor) BLU-9931 (FGFR inhibitor)
DEGRASYN (BCR-ABL inhibitor) DEGRASYN (BCR-ABL inhibitor)
DBEQ (P97 inhibitor) DBEQ (P97 inhibitor)
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor) VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
LINIFANIB (VEGFR inhibitor) LINIFANIB (VEGFR inhibitor)
ML141 (RHO inhibitor) ML141 (RHO inhibitor)
BYL719 (PI3K inhibitor) BYL719 (PI3K inhibitor)
PI-103 (PI3K inhibitor) PI-103 (PI3K inhibitor)
PFI-4 (EPIGENETIC READER DOMAIN inhibitor) PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
ODANACATIB (CYSTEINE PROTEASE inhibitor) ODANACATIB (CYSTEINE PROTEASE inhibitor)
A83-01 (ALK5 inhibitor) A83-01 (ALK5 inhibitor)
タフトシン タフトシン 9063-57-4 C21H40N8O6
SRT 1720 (SIRT1 activator) SRT 1720 (SIRT1 activator)
FK-506 (MTOR inhibitor) FK-506 (MTOR inhibitor)
[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate [oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate 193743-89-4
PFI-3 (EPIGENETIC READER DOMAIN inhibitor) PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
BAY87-2243 (HIF inhibitor) BAY87-2243 (HIF inhibitor)
INDIPLON (GABA RECEPTOR Conditioner) INDIPLON (GABA RECEPTOR Conditioner)
SEMAGACESTAT (GAMMA - SECRETASE Inhibitor) SEMAGACESTAT (GAMMA - SECRETASE Inhibitor)
TG101348 (JAK inhibitor) TG101348 (JAK inhibitor)
PLX4032 (RAF inhibitor) PLX4032 (RAF inhibitor)
ENTOSPLETINIB (SYK inhibitor) ENTOSPLETINIB (SYK inhibitor)
IONOMYCIN (calcium ionophore) IONOMYCIN (calcium ionophore)
PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist) PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist)
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor) SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
EPZ-6438 (E7438) (EZH2 inhibitor) EPZ-6438 (E7438) (EZH2 inhibitor)
SC-514 (IΚB/IKK inhibitor) SC-514 (IΚB/IKK inhibitor)
REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor) REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor) EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
PONATINIB (SRC-ABL inhibitor) PONATINIB (SRC-ABL inhibitor)
ICA 069673 ICA 069673 582323-16-8 C11H6ClF2N3O
BTdCPU BTdCPU 1257423-87-2 C13H8Cl2N4OS
TEDIZOLID (MAO-A inhibitor) TEDIZOLID (MAO-A inhibitor)
PLERIXAFOR (CXCR inhibitor) PLERIXAFOR (CXCR inhibitor)
HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride Cl2H8N2O2
FIPI (PLD1/2 inhibitor) FIPI (PLD1/2 inhibitor)
ABT-199 (BCL-2 inhibitor) ABT-199 (BCL-2 inhibitor)
ポルフィロマイシン ポルフィロマイシン 801-52-5 C16H20N4O5
TIVOZANIB (VEGFR inhibitor) TIVOZANIB (VEGFR inhibitor)
I-BET-762 (GSK525762) (BET inhibitor) I-BET-762 (GSK525762) (BET inhibitor)
BMS-5 (LIMK inhibitor) BMS-5 (LIMK inhibitor)
DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor) DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
SALUBRINAL (PERK inhibitor) SALUBRINAL (PERK inhibitor)
ENZALUTAMIDE (MDV3100) (AR inhibitor) ENZALUTAMIDE (MDV3100) (AR inhibitor)
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor) COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist) BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist)
NECROSTATIN-1 (TNF-ALPHA inhibitor) NECROSTATIN-1 (TNF-ALPHA inhibitor)
SP600125 (JNK inhibitor) SP600125 (JNK inhibitor)
GELDANAMYCIN (HSP90 inhibitor) GELDANAMYCIN (HSP90 inhibitor)
TPA Deficient Plasma TPA Deficient Plasma
AR-A014418 (GSK-3 inhibitor) AR-A014418 (GSK-3 inhibitor)
DALCETRAPIB (CETP inhibitor) DALCETRAPIB (CETP inhibitor)
MI-2 (HISTONE METHYLTRANSFERASE Inhibitor) MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
ML323 (DUB inhibitor) ML323 (DUB inhibitor)
AG14361 (PARP1 inhibitor) AG14361 (PARP1 inhibitor)
IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor) IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
PAC-1 (CASPASE Activator) PAC-1 (CASPASE Activator)
SRT 2104 (SIRT1 activator) SRT 2104 (SIRT1 activator)
ROMIDEPSIN (HDAC inhibitor) ROMIDEPSIN (HDAC inhibitor)
DACOMITINIB (EGFR inhibitor) DACOMITINIB (EGFR inhibitor)
FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor) FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
INH1 (MICROTUBULE ASSOCIATED inhibitor) INH1 (MICROTUBULE ASSOCIATED inhibitor)
RIMONABANT (CANNABINOID RECEPTOR antagonist) RIMONABANT (CANNABINOID RECEPTOR antagonist)
AG1024 (IGF-1R inhibitor) AG1024 (IGF-1R inhibitor)
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