| Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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| Tel: |
821-50328103-801 18930552037 |
| Email: |
3bsc@sina.com |
| Products Intro: |
Product Name:FR 139317;N-[N-[N-[(Hexahydro-1H-azepin-1-yl)carbonyl]-L-leucyl]-1-Methyl-D-tryptophyl]-3-(2-pyridinyl)-D-alanine
CAS:142375-60-8
Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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FR 139317 manufacturers
- FR 139317
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- $2500.00 / 100mg
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2026-01-04
- CAS:142375-60-8
- Min. Order:
- Purity:
- Supply Ability: 10g
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| | FR 139317 Basic information |
| Product Name: | FR 139317 | | Synonyms: | FR 139317;(HEXAHYDRO-1H-AZEPINYL)CARBONYL-LEU-D-(1-ME)-TRP-DPAL;(HEXAHYDRO-1H-AZEPINYL)CARBONYL-LEU-DTRP(ME)-D-ALA(2-PYRIDYL)-OH;2-((1-(Hexahydro-1H-azepinyl)carbonyl)amino-4-methylpentanoyl)-3-(-(1-methyl-1H-indolyl)propionyl)amino-3-(2-pyridyl)propionic acid;D-Alanine, N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl-1-methyl-D-tryptophyl-3-(2-pyridinyl)-;D-Alanine, N-(N-(N-((hexahydro-1H-azepin-1-yl)carbonyl)-L-leucyl)-1-methyl-D-tryptophyl)-3-(2-pyridinyl)-;(2R)-2-[[(2R)-2-[[(2S)-2-(AZEPANE-1-CARBONYLAMINO)-4-METHYLPENTANOYL]AMINO]-3-(1-METHYLINDOL-3-YL)PROPANOYL]AMINO]-3-PYRIDIN-2-YLPROPANOIC ACID;FR139317,CID107810 | | CAS: | 142375-60-8 | | MF: | C33H44N6O5 | | MW: | 604.74 | | EINECS: | | | Product Categories: | | | Mol File: | 142375-60-8.mol |  |
| | FR 139317 Chemical Properties |
| Boiling point | 943.9±65.0 °C(Predicted) | | density | 1.27±0.1 g/cm3(Predicted) | | storage temp. | Desiccate at +4°C | | solubility | Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO | | form | Powder | | pka | 2.68±0.10(Predicted) |
| | FR 139317 Usage And Synthesis |
| Uses | FR 139317 is a novel, potent endothelin ETA receptor antagonist. | | Biological Activity | A highly potent and selective ET A endothelin receptor antagonist (K i values are 1 nM and 7.3 μ M at ET A and ET B subtypes respectively). Active in vivo . | | IC 50 | ETA |
| | FR 139317 Preparation Products And Raw materials |
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