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Recilisib sodium

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Recilisib sodium manufacturers

Recilisib sodium Basic information
Product Name:Recilisib sodium
Synonyms:Ex-Rad;4-[(E)-2-[(4-chlorophenyl)methylsulfonyl]ethenyl]benzoate;4-I(E)-2-[(4-chlorophenyl)methanesulfonyl] ethenyl]benzoate sodium;Brand name: Ex-RAD;ON 01210.Na;ON01210 sodium;ON-01210 sodium
CAS:922139-31-9
MF:C16H12ClNaO4S
MW:360.78
EINECS:
Product Categories:
Mol File:922139-31-9.mol
Recilisib sodium Structure
Recilisib sodium Chemical Properties
Safety Information
MSDS Information
Recilisib sodium Usage And Synthesis
UsesRecilisib sodium (ON 01210) is a radioprotectant, which can activate AKT, PI3K activities in cells[1].
in vivo

Recilisib sodium (500 mg/kg) significantly increases the rate of recovery and differentiation of primitive bone marrow myeloid progenitor cells in mice. Recilisib sodium in combination with radiation reduces CFU numbers in mice, but the Recilisib sodium-treated mice consistently retain a capability to form differentiated colonies. Recilisib sodium treated mice have a progenitor cell population that is never completely depleted by radiation exposure[1].

References[1] Kang AD, et al. ON01210.Na (Ex-RAD) mitigates radiation damage through activation of the AKT pathway. PLoS One. 2013;8(3):e58355. DOI:10.1371/journal.pone.0058355
Recilisib sodium Preparation Products And Raw materials
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