TELENZEPINE 2HCL

Request For Quotation
TELENZEPINE 2HCL Suppliers list
Company Name: Sigma-Aldrich  
Tel: 021-61415566 800-8193336
Email: orderCN@merckgroup.com
Company Name: TargetMol Chemicals Inc.  
Tel: 15002134094
Email: marketing@targetmol.cn
Company Name: Nanjing Jiusinuo Biomedical Technology Co., Ltd.  
Tel: 19822625399
Email: njjsn2023@126.com
Company Name: TargetMol Chemicals Inc.  
Tel: 13564774135
Email: marketing@targetmol.com
Company Name: TargetMol Chemicals Inc.  
Tel: +1-781-999-5354;
Email: support@targetmol.com

TELENZEPINE 2HCL manufacturers

  • Telenzepine
  • Telenzepine pictures
  • $1980.00
  • 2026-04-20
  • CAS:80880-90-6
  • Purity:
  • Supply Ability: 10g
TELENZEPINE 2HCL Basic information
Product Name:TELENZEPINE 2HCL
Synonyms:TELENZEPINE 2HCL;4,9-dihydro-3-methyl-4-[(4-methyl-1-piperazinyl)acetyl]-10h-thieno[3,4-b][1,5]benzodiazepin-10-one dihydrobromide;telenzepine dihydrochloride hydrate;SK-871;1-methyl-10-[2-(4-methylpiperazin-1-yl)acetyl]-5H-thieno[3,4-b][1,5]benzodiazepin-4-one;10H-Thieno[3,4-b][1,5]benzodiazepin-10-one, 4,9-dihydro-3-methyl-4-[2-(4-methyl-1-piperazinyl)acetyl]-;Telenzepine
CAS:80880-90-6
MF:C19H22N4O2S
MW:370.475
EINECS:
Product Categories:
Mol File:80880-90-6.mol
TELENZEPINE 2HCL Structure
TELENZEPINE 2HCL Chemical Properties
Melting point 263-264°
Boiling point 544.7±50.0 °C(Predicted)
density 1.281±0.06 g/cm3(Predicted)
solubility H2O: >10 mg/mL
pka12.48±0.20(Predicted)
form solid
color white
Safety Information
WGK Germany 3
MSDS Information
TELENZEPINE 2HCL Usage And Synthesis
UsesTelenzepine is an antimuscarinic agent with Kis of 0.94 nM (M1 mAChR) and 17.8 nM (M2 mAChR) binding to muscarinic receptors. Telenzepine effectively blocks synaptic transmission promoted by muscarinic or M1 receptor agonists. Thus, Telenzepine can reduce the amplitude of extracellular slow excitatory postsynaptic potentials (EC50=38 nM) and slow inhibitory postsynaptic potentials (EC50=253 nM)[1].
DefinitionChEBI: 1-methyl-10-[2-(4-methyl-1-piperazinyl)-1-oxoethyl]-5H-thieno[3,4-b][1,5]benzodiazepin-4-one is a benzodiazepine.
References[1] Telenzepine. IMGT. DOI:10.1016/0014-2999(89)90741-3
TELENZEPINE 2HCL Preparation Products And Raw materials
Tag:TELENZEPINE 2HCL(80880-90-6) Related Product Information
1-(2-Dimethylaminoethyl)-4-methylpiperazine 1-(4-CHLOROBENZYL)PIPERAZINE N,N-DIMETHYL-2-PIPERAZIN-1-YL-ACETAMIDE 4-Methyl-1-piperazineethanamine N-3-thienylacetamide N-Aminoethylpiperazine TELENZEPINE 2HCL N-Methyl-N-phenyl-2-piperazin-1-ylacetamide N-(2-Amino-ethyl)-benzene-1,2-diamine 3-THIOPHENECARBOXAMIDE 98 1-Piperazineethanamine,N,4-dimethyl-(9CI) N-(2-aminophenyl)-2-(4-methylpiperazin-1-yl)acetamide TELENZEPINE DIHYDROCHLORIDE (4-METHYL-PIPERAZIN-1-YL)-ACETALDEHYDE METHYL-THIOPHEN-3-YLMETHYL-AMINE 3-Amino-4-methylthiophene 2-Piperazin-1-yl-acetamide N1-[2-(Acetylamino)phenyl]acetamide