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| | Ac-Phe-Phe-His-OMe Basic information |
| Product Name: | Ac-Phe-Phe-His-OMe | | Synonyms: | ACETYL-L-PHENYLALANYL-L-PHENYALANYL-L-HISTIDINE METHYL ESTER;TRIPEPTIDE ZAMI 420;zami420;Triletide;N-Acetyl-L-phenylalanyl-L-phenylalanyl-L-histidine methyl ester;L-Histidine, N-acetyl-L-phenylalanyl-L-phenylalanyl-, methyl ester;Ac-Phe-Phe-His-OMe | | CAS: | 62087-96-1 | | MF: | C27H31N5O5 | | MW: | 505.57 | | EINECS: | 263-401-1 | | Product Categories: | | | Mol File: | 62087-96-1.mol |  |
| | Ac-Phe-Phe-His-OMe Chemical Properties |
| Boiling point | 910.0±65.0 °C(Predicted) | | density | 1+-.0.06 g/cm3(Predicted) | | storage temp. | -15°C | | pka | 12.92±0.46(Predicted) |
| | Ac-Phe-Phe-His-OMe Usage And Synthesis |
| Uses | Triletide is a thromboxane A2 antagonist with good oral absorption activity. The biotransformation of Triletide mainly includes the formation of demethyl, deacetyl, demethyl-deacetyl and hydroxy derivatives. The distribution half-life of Triletide is about 1 hour, and the elimination half-life is about 5 hours[1]. | | References | [1] Preliminary human pharmacokinetics of triletide PMID:4059299 |
| | Ac-Phe-Phe-His-OMe Preparation Products And Raw materials |
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