6-BN-cAMP sodium salt

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6-BN-cAMP sodium salt Basic information
Product Name:6-BN-cAMP sodium salt
Synonyms:N6-BENZYLADENOSINE-3',5'-CYCLIC MONOPHOSPHATE SODIUM SALT;6-BN-CAMP, NA;ADENOSINE 3',5'-CYCLIC MONOPHOSPHATE, N6-BENZYL-, SODIUM SALT;n(6)-benzyl-cyclicadenosine5’-monophosphate;n6-benzyladenosine-3’,5’-cyclicmonophosphate(6-bn-camp),sodiumsalt;Adenosine, N-(phenylmethyl)-, cyclic 3',5'-(hydrogen phosphate);[(2R,3R,4R,5R)-2-(2-amino-6-oxo-1H-purin-9-yl)-4-hydroxy-5-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]oxolan-3-yl] 2-(methylamino)benzoate;[(2R,3S,4R,5R)-5-(2-amino-6-oxo-1H-purin-9-yl)-4-hydroxy-2-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]oxolan-3-yl] 2-(methylamino)benzoate
CAS:32115-08-5
MF:C17H18N5O6P
MW:419.33
EINECS:
Product Categories:
Mol File:32115-08-5.mol
6-BN-cAMP sodium salt Structure
6-BN-cAMP sodium salt Chemical Properties
Boiling point 719.8±70.0 °C(Predicted)
density 1.86±0.1 g/cm3(Predicted)
pka1.00±0.60(Predicted)
Safety Information
MSDS Information
6-BN-cAMP sodium salt Usage And Synthesis
Uses6-Bn-cAMP is a site-selective activator of cAMP-dependent protein kinase (PKA) which does not activate Epac. 6-Bn-cAMP increases hydrolytic stability against PDE, esterases, amidases and considerably higher membrane permeability compared to cAMP[1].
References[1] Pepe S, et al. Effects of 8-chloroadenosine 3',5'-monophosphate and N6-benzyl-cyclic adenosine 5'-monophosphate on cell cycle kinetics of HL-60 leukemia cells. Cancer Res. 1991 Dec 1;51(23 Pt 1):6263-7. PMID:1657383
6-BN-cAMP sodium salt Preparation Products And Raw materials
Tag:6-BN-cAMP sodium salt(32115-08-5) Related Product Information
6-BN-cAMP sodium salt 6-Bnz-cAMP sodium salt N6-Benzyladenosine Adenosine 3',5'-cyclic monophosphate sodium salt PROTEIN KINASE A INHIBITOR 14-22 AMIDE, CELL-PERMEABLE, MYRISTOYLATED Sitagliptin