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Mps1-IN-5

Mps1-IN-5 Suppliers list
Company Name: Nanjing Chemlin Chemical Co., Ltd  
Tel: 025-83697070 13770331960
Email: info@chemlin.com.cn
Company Name: BOC Sciences  
Tel: 1-631-485-4226; 16314854226
Email: info@bocsci.com
Company Name: Haoyuan Chemexpress Co., Ltd.  
Tel: 021-58950125
Email: info@chemexpress.com
Company Name: ShangHai Caerulum Pharma Discovery Co., Ltd.  
Tel: 18149758185 18149758185
Email: sales-cpd@caerulumpharma.com
Company Name: Shanghai Lollane Biological Technology Co.,Ltd.  
Tel: 021-52996696,15000506266 15000506266
Email:

Mps1-IN-5 manufacturers

  • Empesertib
  • Empesertib pictures
  • $63.00
  • 2026-07-17
  • CAS:1443763-60-7
  • Purity: 99.40%
  • Supply Ability: 10g
  • Mps1-IN-5
  • Mps1-IN-5 pictures
  • 2025-04-04
  • CAS:1443763-60-7
  • Min. Order: 1KG
  • Purity: 98%
  • Supply Ability: 1ton
Mps1-IN-5 Basic information
Product Name:Mps1-IN-5
Synonyms:CS-2060;BAY-1161909;BAY1161909;Mps1-IN-5;BAY 1161909;Benzeneacetamide, 4-fluoro-N-[4-[2-[[2-methoxy-4-(methylsulfonyl)phenyl]amino][1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]-α-methyl-, (αR)-;BAY-1161909 Empesertib;(Empesertib)BAY1161909;(R)-2-(4-Fluorophenyl)-N-(4-(2-((2-methoxy-4-(methylsulfonyl)phenyl)amino)-[1,2,4]triazolo[1,5-a]pyridin-6-yl)phenyl)propanamide
CAS:1443763-60-7
MF:C29H26FN5O4S
MW:559.62
EINECS:
Product Categories:API
Mol File:1443763-60-7.mol
Mps1-IN-5 Structure
Mps1-IN-5 Chemical Properties
density 1.36±0.1 g/cm3(Predicted)
storage temp. Store at -20°C
solubility DMSO:67.5(Max Conc. mg/mL);120.62(Max Conc. mM)
form Solid
pka13.71±0.70(Predicted)
color White to off-white
Safety Information
MSDS Information
Mps1-IN-5 Usage And Synthesis
UsesEmpesertib (BAY 1161909) is a potent Mps1 inhibitor, with an IC50 of < 1 nM.
IC 50Mps1: 1 nM (IC50)
References[1] SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2
Mps1-IN-5 Preparation Products And Raw materials
Tag:Mps1-IN-5(1443763-60-7) Related Product Information
Mps1-IN-5 BAY-1217389 BAY-1816032 MPI-0479605 [1,2,4]Triazolo[4,3-a]quinoxaline, 8-[5-(difluoromethyl)-3-pyridinyl]-1-(2,3,6,7-tetrahydro-4-oxepinyl)- BAY-2402234