| Company Name: |
BOC Sciences |
| Tel: |
16314854226; +8616314854226 |
| Email: |
inquiry@bocsci.com |
AMASTATIN manufacturers
- Amastatin
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- $2500.00
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2026-05-11
- CAS:67655-94-1
- Purity:
- Supply Ability: 10g
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| | AMASTATIN Basic information |
| Product Name: | AMASTATIN | | Synonyms: | (2S,3R)-3-AMINO-2-HYDROXY-5-METHYLHEXANOYL-VAL-VAL-ASP-OH;[(2S,3R)-3-AMINO-2-HYDROXY-5-METHYLHEXANOYL]-L-VALYL-L-VALYL-L-ASPARTIC ACID;AMASTATIN, STREPTOMYCES SPECIES;AMASTATIN;(AMINO-2-HYDROXY-5-METHYL-HEXANOYL)-L-VALYL-L-VALYL-L-ASPARTIC ACID;N-[(2S,3R)-3-Amino-2-hydroxy-5-methylhexanoyl]-L-Val-L-Val-L-Asp-OH;N-[N-[N-[(2S,3R)-3-Amino-2-hydroxy-5-methyl-1-oxohexyl]-L-valyl]-L-valyl]-L-aspartic acid;[(2S,3R)-3-Amino-2-hydroxy-5-methylhexanoyl]-Val-val-Asp | | CAS: | 67655-94-1 | | MF: | C21H38N4O8 | | MW: | 474.55 | | EINECS: | | | Product Categories: | inhibitor | | Mol File: | 67655-94-1.mol |  |
| | AMASTATIN Chemical Properties |
| Boiling point | 795℃ | | density | 1.228 | | Fp | 435℃ | | form | powder | | pka | 2.865±0.10(predicted) | | color | White |
| Hazard Codes | Xi | | Risk Statements | 36/37/38 | | Safety Statements | 26-36 | | HS Code | 29241900 |
| | AMASTATIN Usage And Synthesis |
| Uses | Amastatin is A slow, tightly bound, competitive inhibitor of aminopeptidase (AP) with an IC50 of 0.54 μg/mL for AP-A[1][2]. | | Definition | ChEBI: A tetrapeptide comprising (2S,3R)-3-amino-2-hydroxy-5-methylhexanoyl, L-valyl, L-valyl and L-aspartic acid units joined in sequence | | References | [1] Aoyagi T, et al. Amastatin, an inhibitor of aminopeptidase A, produced by actinomycetes. J Antibiot (Tokyo). 1978 Jun;31(6):636-8. DOI:10.7164/antibiotics.31.636
[2] Wilkes SH, et al. The slow, tight binding of bestatin and amastatin to aminopeptidases. J Biol Chem. 1985 Oct 25;260(24):13154-62. PMID:2865258 |
| | AMASTATIN Preparation Products And Raw materials |
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