D3-βArr NEW
| Price | $31 | $52 | $113 |
| Package | 5mg | 10mg | 25mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-11-04 |
Product Details
| Product Name: D3-βArr | CAS No.: 662164-09-2 |
| Purity: 98.82% | Supply Ability: 10g |
| Release date: 2025/11/04 |
Product Introduction
Bioactivity
| Name | D3-βArr |
| Description | D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct TSHR activation. |
| In vitro | D3-βArr stimulated β-Arr 1 translocation with an efficacy threefold greater than TSH. The EC50 for β-Arr 1 translocation by D3-βArr was 11.6 μM. D3-βArr (10 μM) increased the efficacy of TSH in the translocation of β-Arr 1 at a maximum of 5.1-fold over TSH alone. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | 10% DMSO+40% PEG300+5% Tween 80+45% Saline : 4 mg/mL (12 mM), Sonication is recommended. DMSO : 100 mg/mL (299.91 mM), Sonication is recommended. |
| Keywords | TSHReceptor | TSH Receptor | thyrotropin receptor (TSHR) | Thyrotropin receptor | Thyroid-stimulating hormone Receptor | NCGC-00379308 | NCGC 00379308 | Inhibitor | inhibit | D3-βArr | D-3-βArr | D3βArr | D3-betaArr | D3-bArr | D3 βArr |
| Inhibitors Related | Teprotumumab | TSHR antagonist S37 | ML224 | VA-K-14 hydrochloride | NCATS-SM4420 | Org41841 | K1-70 | ML-109 | NCGC00229600 |
| Related Compound Libraries | Osteogenesis Compound Library | Nuclear Receptor Compound Library | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Endocrinology-Hormone Compound Library | NO PAINS Compound Library | Bioactive Compounds Library Max | GPCR Compound Library | Anti-Cancer Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, MA
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